SCHEMBL8890958

SCHEMBL8890958

Clc1nc(Nc2ccccc2)c2cc(-c3ccccc3)ccc2n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 4/20 0.53
RAF1 P04049 3/20 0.53
EGLN1 Q9GZT9 1/20 0.52
LMNA P02545 4/20 0.50
CYP1A2 P05177 4/20 0.50
CYP3A4 P08684 4/20 0.50
MAPK1 P28482 3/20 0.50
HIF1A Q16665 2/20 0.50
MEN1 O00255 5/20 0.49
KMT2A Q03164 5/20 0.49
ABCG2 Q9UNQ0 4/20 0.49
TRIM58 Q8NG06 1/20 0.49
USP2 O75604 3/20 0.48
TSHR P16473 3/20 0.48
CYP2C19 P33261 3/20 0.48
CLK4 Q9HAZ1 3/20 0.48
CYP2C9 P11712 1/20 0.48
HSD17B10 Q99714 1/20 0.48
PDE5A O76074 4/20 0.48
CYP2D6 P10635 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8897789 0.83 NPY5R (0.66) BRAFRAF1EGLN1LMNACYP1A2
SCHEMBL2257238 0.80 NPY5R (0.66) MAPK1MEN1KMT2AABCG2CLK4
SCHEMBL30960995 0.80 NPY5R (0.66) MAPK1MEN1KMT2AABCG2CLK4
SCHEMBL6039347 0.78 EGFR (0.65) BRAFLMNACYP1A2CYP3A4MAPK1
SCHEMBL8899763 0.77 KDM4E (0.50) LMNACYP1A2MEN1KMT2ATRIM58
SCHEMBL15051337 0.77 BRAF (0.84) BRAFRAF1LMNACYP1A2CYP3A4
SCHEMBL8898615 0.76 ABCG2 (0.71) KMT2AABCG2
SCHEMBL19639039 0.76 KDM4E (0.71) LMNAMAPK1MEN1KMT2ATRIM58
SCHEMBL17367223 0.76 KDM4E (0.71) LMNAMAPK1MEN1KMT2ATRIM58
SCHEMBL29992999 0.76 KDM4E (0.71) LMNAMAPK1MEN1KMT2ATRIM58

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020822-A1 QUINAZOLIN-2,4-DIAZIRINES AS NPY RECEPTOR ANTAGONIST NOVARTIS AG (CH) 1997-06-12 WO disclosed