SCHEMBL8897789

SCHEMBL8897789

c1ccc(Nc2nc(Nc3ccccc3)c3cc(-c4ccccc4)ccc3n2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 6/20 0.66
TRIM58 Q8NG06 1/20 0.61
RAF1 P04049 3/20 0.55
BRAF P15056 3/20 0.55
LMNA P02545 3/20 0.54
CYP1A2 P05177 3/20 0.54
CYP3A4 P08684 3/20 0.54
MAPK1 P28482 2/20 0.54
HIF1A Q16665 1/20 0.54
EGLN1 Q9GZT9 1/20 0.53
ADRB2 P07550 1/20 0.51
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
ABCG2 Q9UNQ0 2/20 0.50
USP2 O75604 2/20 0.49
TSHR P16473 2/20 0.49
CYP2C19 P33261 2/20 0.49
CLK4 Q9HAZ1 2/20 0.49
CYP2C9 P11712 1/20 0.49
HSD17B10 Q99714 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8901062 0.86 NPY5R (0.84) NPY5RLMNACYP1A2CYP3A4MEN1
Hydrochloric Acid SCHEMBL8900034 0.84 NPY5R (0.81) NPY5RLMNACYP1A2CYP3A4MAPK1
SCHEMBL21500678 0.83 ADRB2 (0.69) NPY5RTRIM58MAPK1ADRB2MEN1
SCHEMBL8890958 0.83 BRAF (0.53) TRIM58RAF1BRAFLMNACYP1A2
SCHEMBL8900516 0.81 NPY5R (0.77) NPY5RTRIM58BRAFLMNACYP1A2
Hydrochloric Acid SCHEMBL8890109 0.80 NPY5R (0.76) NPY5RTRIM58BRAFLMNACYP1A2
SCHEMBL2591063 0.80 NPY5R (1.00) NPY5RMAPK1MEN1KMT2AABCG2
Hydrochloric Acid SCHEMBL6039677 0.78 NPY5R (0.96) NPY5RMAPK1MEN1KMT2AABCG2
SCHEMBL15051337 0.78 BRAF (0.84) RAF1BRAFLMNACYP1A2CYP3A4
SCHEMBL8893267 0.78 NPY5R (0.60) NPY5RSLC2A1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020822-A1 QUINAZOLIN-2,4-DIAZIRINES AS NPY RECEPTOR ANTAGONIST NOVARTIS AG (CH) 1997-06-12 WO claimed
WO-1997020822-A1 QUINAZOLIN-2,4-DIAZIRINES AS NPY RECEPTOR ANTAGONIST NOVARTIS AG (CH) 1997-06-12 WO disclosed