SCHEMBL8891361

SCHEMBL8891361

CC[N+](CC)(CCC(=O)N1C[C@H]2[C@@H](C1Br)C(c1ccccc1)(c1ccccc1)C[C@@H](O)[C@]2(O)c1cc(OC)ccc1OC)Cc1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.34
KDM4E B2RXH2 2/20 0.34
GAA P10253 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
SIGMAR1 Q99720 2/20 0.33
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
POLB P06746 1/20 0.32
TACR1 P25103 1/20 0.31
GRIN2B Q13224 1/20 0.31
EDNRA P25101 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8890176 0.89 KDM4E (0.34) ALDH1A1KDM4EGAATDP1SIGMAR1
Bromide SCHEMBL8891355 0.86 ALDH1A1 (0.38) ALDH1A1KDM4EGAATDP1SIGMAR1
SCHEMBL8890828 0.81 TACR1 (0.33) TACR1GRIN2B
Bromide SCHEMBL8890170 0.75 ALDH1A1 (0.37) ALDH1A1KDM4EGAATDP1SIGMAR1
SCHEMBL8891331 0.71 TACR1 (0.39) KMT2AMEN1TACR1GRIN2B
SCHEMBL8892577 0.69 TACR1 (0.39) GAASIGMAR1KMT2AMEN1TACR1
Bromide SCHEMBL8890180 0.69 TACR1 (0.38) ALDH1A1KDM4EGAATDP1TACR1
Bromide SCHEMBL8891366 0.69 TACR1 (0.37) ALDH1A1KDM4EGAATDP1TACR1
SCHEMBL8891902 0.68 SIGMAR1 (0.39) ALDH1A1KDM4EGAASIGMAR1KMT2A
Bromide SCHEMBL8891352 0.68 TACR1 (0.41) ALDH1A1KDM4EGAATDP1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997005110-A1 PERHYDROISOINDOLE DERIVATIVES AS SUBSTANCE P AND NEUROKININE A ANTAGONISTS RHONE-POULENC RORER S.A. (FR) 1997-02-13 WO claimed
WO-1997005110-A1 PERHYDROISOINDOLE DERIVATIVES AS SUBSTANCE P AND NEUROKININE A ANTAGONISTS RHONE-POULENC RORER S.A. (FR) 1997-02-13 WO disclosed