SCHEMBL8891646

SCHEMBL8891646

COCCc1ccc(Nc2nc(Nc3ccc(C(N)=O)cc3)c3ccccc3n2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 1/20 0.55
NPY5R Q15761 8/20 0.54
KDM1A O60341 1/20 0.52
PDE5A O76074 1/20 0.49
ABCC1 P33527 1/20 0.49
ABCG2 Q9UNQ0 1/20 0.49
LRRK2 Q5S007 1/20 0.48
KDM4E B2RXH2 2/20 0.48
ALDH1A1 P00352 2/20 0.48
GAA P10253 2/20 0.48
MAPT P10636 2/20 0.48
HPGD P15428 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
SLC2A1 P11166 1/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
CYP1A2 P05177 1/20 0.47
POLB P06746 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8890748 0.88 NPY5R (0.67) PIN1NPY5RSLC2A1MERTK
SCHEMBL8890470 0.84 NPY5R (0.70) PIN1NPY5RKDM1AABCC1ABCG2
SCHEMBL8889582 0.84 NPY5R (0.76) NPY5RABCC1ABCG2ALDH1A1MAPT
SCHEMBL8889731 0.81 NPY5R (0.59) PIN1NPY5RKDM4EALDH1A1GAA
SCHEMBL8891586 0.80 NPY5R (0.65) NPY5RPDE5AABCG2KDM4EALDH1A1
Hydrochloric Acid SCHEMBL8901384 0.79 NPY5R (0.64) NPY5RPDE5AABCG2KDM4EALDH1A1
SCHEMBL8889728 0.75 NPY5R (0.70) NPY5RKDM4EALDH1A1GAAMAPT
SCHEMBL8899488 0.75 NPY5R (0.69) NPY5RSLC2A1MERTK
SCHEMBL8891004 0.75 NPY5R (0.62) PIN1NPY5RLRRK2PDE4B
Hydrochloric Acid SCHEMBL8900880 0.74 NPY5R (0.68) NPY5RSLC2A1POLBMERTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020822-A1 QUINAZOLIN-2,4-DIAZIRINES AS NPY RECEPTOR ANTAGONIST NOVARTIS AG (CH) 1997-06-12 WO claimed