SCHEMBL8890470

SCHEMBL8890470

NC(=O)c1ccc(Nc2nc(Nc3ccccc3)c3ccccc3n2)cc1

nearest known ligand 0.70

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 9/20 0.70
PIN1 Q13526 2/20 0.66
AURKA O14965 1/20 0.62
JAK2 O60674 1/20 0.62
AURKB Q96GD4 1/20 0.62
KDM1A O60341 1/20 0.61
LRRK2 Q5S007 1/20 0.60
MERTK Q12866 1/20 0.57
ABCC1 P33527 1/20 0.56
ABCG2 Q9UNQ0 1/20 0.56
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
SIRT5 Q9NXA8 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8891646 0.84 PIN1 (0.55) NPY5RPIN1AURKAJAK2AURKB
SCHEMBL2591063 0.84 NPY5R (1.00) NPY5RPIN1AURKAMERTKABCG2
SCHEMBL9938046 0.84 ABCG2 (0.80) KDM1AABCC1ABCG2MEN1KMT2A
Benzene SCHEMBL28899784 0.83 MAPT (0.61) PIN1KDM1ALRRK2ABCC1ABCG2
SCHEMBL4147023 0.83 MAPT (0.61) PIN1KDM1ALRRK2ABCC1ABCG2
Hydrochloric Acid SCHEMBL6039677 0.82 NPY5R (0.96) NPY5RPIN1AURKAABCG2MEN1
SCHEMBL8890734 0.81 NPY5R (0.81) NPY5RMERTKABCG2MEN1KMT2A
Hydrochloric Acid SCHEMBL8900449 0.81 NPY5R (0.81) NPY5RPIN1KDM1AMERTKMEN1
Hydrochloric Acid SCHEMBL8889510 0.80 NPY5R (0.79) NPY5RMERTKABCG2MEN1KMT2A
SCHEMBL8898077 0.80 NPY5R (0.84) NPY5RMERTKABCG2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020822-A1 QUINAZOLIN-2,4-DIAZIRINES AS NPY RECEPTOR ANTAGONIST NOVARTIS AG (CH) 1997-06-12 WO claimed