SCHEMBL8891774

SCHEMBL8891774

COc1ccc(C[C@H](C[C@H](O)[C@@H](N)Cc2ccc(OC)cc2)C(=O)O)cc1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.56
PPARG P37231 2/20 0.49
KMT2A Q03164 1/20 0.48
SLC6A4 P31645 1/20 0.47
SLC1A3 P43003 1/20 0.47
SLC1A2 P43004 1/20 0.47
SLC1A1 P43005 1/20 0.47
ANPEP P15144 1/20 0.46
ERAP2 Q6P179 1/20 0.46
PPARA Q07869 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C19 P33261 1/20 0.45
GRIK1 P39086 1/20 0.45
GRIK2 Q13002 1/20 0.45
LTA4H P09960 1/20 0.44
POLB P06746 1/20 0.44
TPH1 P17752 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8891766 1.00 LDHA (0.56) LDHAPPARGKMT2ASLC6A4SLC1A3
SCHEMBL7439269 0.96 SLC1A3 (0.54) LDHAPPARGKMT2ASLC1A3SLC1A2
SCHEMBL8893679 0.96 SLC1A3 (0.54) LDHAPPARGKMT2ASLC1A3SLC1A2
SCHEMBL8893674 0.96 SLC1A3 (0.54) LDHAPPARGKMT2ASLC1A3SLC1A2
SCHEMBL7439274 0.96 SLC1A3 (0.54) LDHAPPARGKMT2ASLC1A3SLC1A2
SCHEMBL8892841 0.95 LDHA (0.51) LDHAPPARGKMT2ASLC6A4SLC1A3
SCHEMBL8892836 0.95 LDHA (0.51) LDHAPPARGKMT2ASLC6A4SLC1A3
SCHEMBL8895252 0.91 TAAR1 (0.49) LDHAPPARGSLC6A4SLC1A3SLC1A2
SCHEMBL8895260 0.91 TAAR1 (0.49) LDHAPPARGSLC6A4SLC1A3SLC1A2
SCHEMBL8893456 0.89 LTA4H (0.61) LDHAPPARGSLC1A3SLC1A2SLC1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5643878-A TREATMENT OF RETROVIRAL DISEASES LIKE AIDS CIBA-GEIGY CORPORATION (US) 1997-07-01 US disclosed
EP-0618222-A2 Dipeptid derivatives of 5-amino-4-hydroxy-hexanoic acid CIBA-GEIGY AG (CH) 1994-10-05 EP disclosed