SCHEMBL8891906

SCHEMBL8891906

O=C(Nc1c(Cl)cncc1Cl)c1cccc(CCc2ccccn2)c1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.60
GAA P10253 1/20 0.60
ALDH1A1 P00352 1/20 0.53
PDE4D Q08499 9/20 0.47
PDE4A P27815 8/20 0.47
PDE4B Q07343 8/20 0.47
PDE4C Q08493 8/20 0.47
HSD11B1 P28845 1/20 0.44
MAPT P10636 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
TYK2 P29597 1/20 0.43
CYP2B6 P20813 1/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8890145 0.79 PDE4D (0.61) KDM4EGAAALDH1A1PDE4DPDE4A
SCHEMBL8892009 0.77 PDE4D (0.55) KDM4EPDE4DPDE4APDE4BPDE4C
SCHEMBL8891655 0.77 PDE4B (0.70) PDE4DPDE4APDE4BPDE4CCYP2B6
SCHEMBL8888975 0.74 PDE4D (0.70) PDE4DPDE4APDE4BPDE4CCYP2B6
SCHEMBL4662144 0.74 KDM4E (0.54) KDM4EGAAALDH1A1HSD11B1MAPT
SCHEMBL3237987 0.73 TYK2 (0.60) PDE4DPDE4APDE4BPDE4CTYK2
SCHEMBL4037514 0.72 PDE4D (0.56) GAAPDE4DPDE4APDE4BPDE4C
SCHEMBL8891135 0.71 PDE4D (0.52) KDM4EPDE4DPDE4APDE4BPDE4C
SCHEMBL8891532 0.70 PDE4D (0.66) PDE4DPDE4APDE4BPDE4CCYP2B6
SCHEMBL9128209 0.69 CYP1A2 (0.56) KDM4EGAAALDH1A1MAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997003967-A1 SUBSTITUTED AROMATIC COMPOUNDS AND THEIR PHARMACEUTICAL USE RHONE-POULENC RORER LIMITED (GB) 1997-02-06 WO claimed
WO-1997003967-A1 SUBSTITUTED AROMATIC COMPOUNDS AND THEIR PHARMACEUTICAL USE RHONE-POULENC RORER LIMITED (GB) 1997-02-06 WO disclosed