SCHEMBL8892643

SCHEMBL8892643

COC(=O)C(C[C@H](NC(=O)[C@H](Cc1ccc(Cl)cc1)NC(=O)[C@@H](CCSC)NC(=O)[C@H](N)Cc1c[nH]c2ccccc12)C(N)=O)C(=O)OC

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 3/20 0.54
CCKAR P32238 1/20 0.54
NPY1R P25929 3/20 0.49
NPY2R P49146 3/20 0.49
NPY4R P50391 3/20 0.49
CTSC P53634 1/20 0.49
IL1RN P18510 2/20 0.48
ERAP2 Q6P179 2/20 0.48
ERAP1 Q9NZ08 1/20 0.48
GHSR Q92847 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8894358 0.94 CCKBR (0.59) CCKBRCCKARCTSCGHSR
SCHEMBL8893123 0.93 CCKBR (0.56) CCKBRCCKARNPY1RNPY2RNPY4R
SCHEMBL8895429 0.93 IL1RN (0.54) NPY1RNPY2RNPY4RIL1RNERAP2
SCHEMBL8894510 0.93 IL1RN (0.54) NPY1RNPY2RNPY4RIL1RNERAP2
SCHEMBL8892946 0.93 CTSC (0.55) CCKBRCCKARNPY1RNPY2RNPY4R
SCHEMBL8894530 0.92 ECE1 (0.53) IL1RNERAP2ERAP1GHSR
SCHEMBL8894394 0.88 CCKBR (0.59) CCKBRCCKARNPY1RNPY2RNPY4R
SCHEMBL8892706 0.87 ECE1 (0.57) IL1RNERAP2ERAP1GHSR
SCHEMBL8893522 0.86 ECE1 (0.59) IL1RNERAP2ERAP1GHSR
SCHEMBL8894507 0.86 ECE1 (0.59) IL1RNERAP2ERAP1GHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5661128-A TREATING CANCER MERCK & CO. INC. (US) 1997-08-26 US claimed
US-5661128-A TREATING CANCER MERCK & CO. INC. (US) 1997-08-26 US disclosed
WO-1996010037-A1 PEPTIDE INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1996-04-04 WO disclosed