SCHEMBL8892709

SCHEMBL8892709

CNc1cc(-n2ccc3ccccc32)cc(C)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BIRC5 O15392 1/20 0.45
NOS3 P29474 1/20 0.43
NOS2 P35228 1/20 0.43
PRKD3 O94806 1/20 0.37
PRKCG P05129 1/20 0.37
PRKCB P05771 1/20 0.37
PRKCA P17252 1/20 0.37
PRKACA P17612 1/20 0.37
PRKACG P22612 1/20 0.37
PRKACB P22694 1/20 0.37
PRKCH P24723 1/20 0.37
PRKCI P41743 1/20 0.37
PRKCE Q02156 1/20 0.37
PRKCQ Q04759 1/20 0.37
PRKCZ Q05513 1/20 0.37
PRKCD Q05655 1/20 0.37
PRKD1 Q15139 1/20 0.37
CDC7 O00311 1/20 0.37
CDK2 P24941 1/20 0.37
ROCK1 Q13464 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8893532 0.87 BIRC5 (0.53) BIRC5PRKD3PRKCGPRKCBPRKCA
SCHEMBL10153905 0.76 BIRC5 (0.64) BIRC5PRKD3PRKCGPRKCBPRKCA
SCHEMBL5216431 0.75 BIRC5 (0.55) BIRC5PRKD3PRKCGPRKCBPRKCA
SCHEMBL28580892 0.75 CDC7 (0.49) BIRC5PRKD3PRKCGPRKCBPRKCA
SCHEMBL9377416 0.75 CDK2 (0.42) BIRC5PRKD3PRKCGPRKCBPRKCA
Dimethylamine SCHEMBL5608192 0.73 BIRC5 (0.61) BIRC5PRKD3PRKCGPRKCBPRKCA
SCHEMBL9377830 0.72 BIRC5 (0.42) BIRC5PRKD3PRKCGPRKCBPRKCA
SCHEMBL13105711 0.72 BIRC5 (0.61) BIRC5PRKD3PRKCGPRKCBPRKCA
Iodide SCHEMBL8894187 0.71 BIRC5 (0.41) BIRC5PRKD3PRKCGPRKCBPRKCA
SCHEMBL4426563 0.70 BIRC5 (0.67) BIRC5PRKD3PRKCGPRKCBPRKCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5654298-A QUARTERNARY SALTS OF 4-AMINO-SUBSTITUTED PYRIDINES; MODULATORS OF THE SINOATRIAL NODE; CARDIOTONIC AND BRADYCARDIA AGENTS; IMPERIAL CHEMICAL INDUSTRIES (GB) 1997-08-05 US disclosed
EP-0453197-B1 Amine derivatives ICI PLC (GB) 1994-06-15 EP disclosed
EP-0453197-A1 Amine derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-10-23 EP disclosed