SCHEMBL8893573

SCHEMBL8893573

NC(=S)c1ccc(N2CC(C(=O)N[C@H](Cc3ccccc3)C(=O)O)OC2=O)cc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.48
KMT2A Q03164 2/20 0.42
LMNA P02545 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CAPN1 P07384 3/20 0.39
POLB P06746 3/20 0.39
CA2 P00918 2/20 0.39
CA1 P00915 1/20 0.39
GRM2 Q14416 1/20 0.38
PTPN1 P18031 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NAALAD2 Q9Y3Q0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7462123 0.90 ADORA2A (0.48) ADORA2AKMT2ALMNATDP1CAPN1
SCHEMBL27505326 0.88 ADORA2A (0.43) ADORA2ATDP1CAPN1POLB
SCHEMBL27563356 0.83 ADORA2A (0.48) ADORA2AKMT2ALMNATDP1POLB
SCHEMBL7457111 0.83 ADORA2A (0.48) ADORA2AKMT2ALMNATDP1POLB
SCHEMBL7463401 0.83 ITGB3 (0.45) ADORA2ACA2CA1NAALAD2
SCHEMBL8892198 0.81 ADORA2A (0.47) ADORA2AKMT2ALMNATDP1POLB
SCHEMBL7462112 0.80 ADORA2A (0.54) ADORA2AKMT2ACA2
SCHEMBL7457527 0.79 ADORA2A (0.43) ADORA2A
SCHEMBL8893137 0.78 ADORA2A (0.49) ADORA2AKMT2ATDP1MEN1
SCHEMBL7456296 0.77 PRSS1 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5614535-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-03-25 US disclosed