SCHEMBL8893663

SCHEMBL8893663

O=C(O)c1cc2ccccc2cc1NC(=O)C(F)(F)F

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.64
GRIK1 P39086 2/20 0.58
MAPT P10636 5/20 0.57
GFER P55789 1/20 0.57
NGLY1 Q96IV0 1/20 0.57
ABCC1 P33527 1/20 0.55
HSD17B10 Q99714 2/20 0.51
KDM4E B2RXH2 2/20 0.51
ALDH1A1 P00352 2/20 0.51
HPGD P15428 2/20 0.51
AKR1C3 P42330 1/20 0.51
AKR1C2 P52895 1/20 0.51
AKR1C1 Q04828 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
PKM P14618 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
IDO1 P14902 1/20 0.46
HDAC1 Q13547 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL432229 0.80 KCNK2 (0.55) GRIK1MAPTHSD17B10ALDH1A1HPGD
SCHEMBL4311266 0.78 PTPN1 (1.00) PTPN1GRIK1MAPTGFERNGLY1
SCHEMBL5860670 0.78 PTPN1 (0.70) PTPN1GRIK1MAPTGFERNGLY1
SCHEMBL12368149 0.76 MAPT (0.60) MAPTHSD17B10KDM4EALDH1A1HPGD
SCHEMBL1893876 0.75 KCNK2 (0.57) PTPN1GRIK1MAPTHSD17B10KDM4E
SCHEMBL9743950 0.75 GRIK1 (0.56) GRIK1MAPTALDH1A1MEN1KMT2A
SCHEMBL2841346 0.75 PTPN1 (0.66) PTPN1GRIK1MAPTGFERNGLY1
SCHEMBL30694140 0.75 SMN1; SMN2 (0.39) PTPN1GRIK1MAPTHSD17B10KDM4E
SCHEMBL16198286 0.74 KDM4E (0.64) HSD17B10KDM4EALDH1A1AKR1C3AKR1C2
SCHEMBL8550609 0.74 GRIK1 (0.56) GRIK1GFERMEN1KMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997014685-A1 PYRIMIDINE DERIVATIVES GYÓGYSZERKUTATÓ INTÉZET KFT (HU) 1997-04-24 WO disclosed