SCHEMBL8898845

SCHEMBL8898845

COc1cccc2c(Nc3ccc(Cl)cc3)nc(Nc3ccc(C(NC(C)=O)OC)cc3)nc12

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 3/20 0.41
EGFR P00533 1/20 0.39
KDR P35968 1/20 0.39
BRAF P15056 1/20 0.39
TNKS O95271 1/20 0.37
TNKS2 Q9H2K2 1/20 0.37
PARP2 Q9UGN5 1/20 0.37
TNF P01375 1/20 0.36
ALK Q9UM73 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
KMT2A Q03164 1/20 0.36
SLC2A1 P11166 1/20 0.36
BRD4 O60885 1/20 0.35
BRD2 P25440 1/20 0.35
BRD3 Q15059 1/20 0.35
AGPAT2 O15120 2/20 0.35
ABCG2 Q9UNQ0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8905477 0.99 NPY5R (0.40) NPY5REGFRKDRBRAFTNKS
SCHEMBL8893955 0.80 NPY5R (0.40) NPY5REGFRKDRTNKSTNKS2
SCHEMBL8891133 0.77 NPY5R (0.46) NPY5RKDRTNKSTNKS2PARP2
SCHEMBL8900353 0.77 NPY5R (0.49) NPY5RMEN1ALDH1A1POLBKMT2A
SCHEMBL8893944 0.76 KMT2A (0.46) NPY5RMEN1ALDH1A1POLBKMT2A
Hydrochloric Acid SCHEMBL8905468 0.75 KMT2A (0.45) NPY5RMEN1ALDH1A1POLBKMT2A
SCHEMBL8890323 0.74 NPY5R (0.45) NPY5REGFRKDRTNF
Hydrochloric Acid SCHEMBL8890553 0.73 NPY5R (0.44) NPY5REGFRTNFSLC2A1
SCHEMBL8900365 0.73 SLC2A1 (0.49) NPY5RMEN1ALDH1A1KMT2ASLC2A1
Hydrochloric Acid SCHEMBL8892373 0.73 EGFR (0.49) EGFRKDRTNKSTNKS2PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020822-A1 QUINAZOLIN-2,4-DIAZIRINES AS NPY RECEPTOR ANTAGONIST NOVARTIS AG (CH) 1997-06-12 WO claimed