SCHEMBL8894627

SCHEMBL8894627

COC(=O)CC(=O)NS(=O)(=O)c1c(-c2ccccc2)noc1C

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.55
NR4A2 P43354 1/20 0.55
ALDH1A1 P00352 6/20 0.47
MT-CO2 P00403 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
GAA P10253 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
PKM P14618 2/20 0.45
NR3C1 P04150 1/20 0.44
NR3C2 P08235 1/20 0.44
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
TSHR P16473 2/20 0.43
PTGS1 P23219 1/20 0.43
POLB P06746 1/20 0.43
ALOX15 P16050 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8896453 0.89 PTGS2 (0.54) PTGS2NR4A2ALDH1A1MT-CO2NPSR1
SCHEMBL6990229 0.88 PTGS2 (0.69) PTGS2NR4A2ALDH1A1MT-CO2NPSR1
SCHEMBL8895853 0.83 PTGS2 (0.52) PTGS2NR4A2ALDH1A1MT-CO2NPSR1
SCHEMBL5071833 0.83 PTGS2 (0.80) PTGS2NR4A2ALDH1A1MT-CO2NPSR1
SCHEMBL8921742 0.80 PTGS2 (0.49) PTGS2NR4A2ALDH1A1MT-CO2NPSR1
SCHEMBL8897672 0.80 PTGS2 (0.49) PTGS2NR4A2ALDH1A1MT-CO2NPSR1
SCHEMBL8911333 0.79 ALDH1A1 (0.53) PTGS2NR4A2ALDH1A1MT-CO2NPSR1
SCHEMBL10154022 0.77 ALDH1A1 (0.53) PTGS2NR4A2ALDH1A1MT-CO2NPSR1
SCHEMBL5073546 0.76 PTGS2 (0.76) PTGS2NR4A2ALDH1A1MT-CO2NPSR1
SCHEMBL5142318 0.74 PTGS2 (0.80) PTGS2NR4A2ALDH1A1MT-CO2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997038986-A1 SUBSTITUTED BENZENESULFONAMIDE DERIVATIVES AS PRODRUGS OF COX-2 INHIBITORS G.D. SEARLE & CO. (US) 1997-10-23 WO disclosed