SCHEMBL8894968

SCHEMBL8894968

CC(=O)NS(=O)(=O)n1cc(C(F)(F)F)nc1-c1cccnc1C

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.55
PTGS1 P23219 2/20 0.38
USP1 O94782 1/20 0.37
PDE2A O00408 1/20 0.37
PDE10A Q9Y233 1/20 0.37
GPBAR1 Q8TDU6 1/20 0.36
TGFBR1 P36897 1/20 0.36
PKM P14618 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5069859 0.81 PTGS2 (0.72) PTGS2PTGS1
SCHEMBL27421541 0.74 PTGS2 (0.59) PTGS2PTGS1
SCHEMBL8896836 0.74 PTGS2 (0.53) PTGS2PTGS1
SCHEMBL8346351 0.73 PTGS2 (0.50) PTGS2PTGS1USP1PDE2APDE10A
SCHEMBL8346344 0.72 PTGS2 (0.55) PTGS2PTGS1USP1PKM
SCHEMBL5594051 0.71 PTGS2 (1.00) PTGS2PTGS1
Sulfamide SCHEMBL4639044 0.71 PTGS2 (0.81) PTGS2PTGS1
SCHEMBL5069869 0.71 PTGS2 (0.66) PTGS2PTGS1
SCHEMBL215052 0.70 PTGS2 (1.00) PTGS2PTGS1
Benzenesulfonamide SCHEMBL7048970 0.68 PTGS2 (0.62) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997038986-A1 SUBSTITUTED BENZENESULFONAMIDE DERIVATIVES AS PRODRUGS OF COX-2 INHIBITORS G.D. SEARLE & CO. (US) 1997-10-23 WO disclosed