SCHEMBL8896836

SCHEMBL8896836

CC(=O)NS(=O)(=O)n1cc(C(F)(F)F)nc1-c1cncc(C)c1

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.53
KCNT1 Q5JUK3 1/20 0.38
PTGS1 P23219 5/20 0.37
PIK3CG P48736 2/20 0.35
PIK3CB P42338 1/20 0.35
SLC22A12 Q96S37 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8905206 0.83 PTGS2 (0.53) PTGS2PTGS1
SCHEMBL5069858 0.79 PTGS2 (0.72) PTGS2PTGS1
SCHEMBL8894968 0.74 PTGS2 (0.55) PTGS2PTGS1
SCHEMBL27444815 0.73 PTGS2 (0.59) PTGS2PTGS1
SCHEMBL5071016 0.71 PTGS2 (0.66) PTGS2PTGS1
SCHEMBL8346615 0.70 PTGS2 (0.50) PTGS2PTGS1
SCHEMBL8348990 0.70 PTGS2 (0.54) PTGS2PTGS1SLC22A12
SCHEMBL3246331 0.69 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL212333 0.68 PTGS2 (1.00) PTGS2PTGS1
Sulfamide SCHEMBL4638575 0.68 PTGS2 (0.80) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997038986-A1 SUBSTITUTED BENZENESULFONAMIDE DERIVATIVES AS PRODRUGS OF COX-2 INHIBITORS G.D. SEARLE & CO. (US) 1997-10-23 WO disclosed