SCHEMBL8895852

SCHEMBL8895852

COC(=O)CC[C@H]1CC[C@H](N2CCN(c3ccc4c(c3)CCN(C(=O)C(F)(F)F)CC4)S2(=O)=O)CC1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.39
ESR2 Q92731 3/20 0.39
USP30 Q70CQ3 6/20 0.33
HDAC6 Q9UBN7 1/20 0.32
TMEM97 Q5BJF2 2/20 0.31
SIGMAR1 Q99720 2/20 0.31
ABHD6 Q9BV23 1/20 0.31
DRD2 P14416 1/20 0.30
DRD3 P35462 1/20 0.30
PDE4B Q07343 1/20 0.30
PDE4D Q08499 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8895858 1.00 ESR1 (0.39) ESR1ESR2USP30HDAC6TMEM97
SCHEMBL8562237 0.81 ESR1 (0.39) ESR1ESR2HDAC6ABHD6PDE4B
SCHEMBL8562233 0.81 ESR1 (0.39) ESR1ESR2HDAC6ABHD6PDE4B
SCHEMBL8567428 0.80 ESR1 (0.40) ESR1ESR2USP30HDAC6ABHD6
SCHEMBL8567424 0.80 ESR1 (0.40) ESR1ESR2USP30HDAC6ABHD6
SCHEMBL8564189 0.80 ESR1 (0.41) ESR1ESR2HDAC6TMEM97SIGMAR1
SCHEMBL8564198 0.80 ESR1 (0.41) ESR1ESR2HDAC6TMEM97SIGMAR1
SCHEMBL8562057 0.79 ESR1 (0.38) ESR1ESR2HDAC6TMEM97SIGMAR1
SCHEMBL8561418 0.79 ESR1 (0.41) ESR1ESR2HDAC6TMEM97SIGMAR1
SCHEMBL8568715 0.79 F10 (0.39) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5612335-A ANTICOAGULANTS; COMBATING/PREVENTING DISEASES WHERE CELL AGGREGATES OCCUR OR CELL-MATRIX INTERACTIONS PLAY A PART KARL THOMAE GMBH (DE) 1997-03-18 US disclosed