SCHEMBL8562233

SCHEMBL8562233

COC(=O)CC[C@H]1CC[C@H](n2ccn(-c3ccc4c(c3)CCN(C(=O)C(F)(F)F)CC4)c2=O)CC1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.39
ESR2 Q92731 3/20 0.39
HDAC6 Q9UBN7 1/20 0.32
ABHD6 Q9BV23 1/20 0.31
LPAR5 Q9H1C0 1/20 0.31
GPR119 Q8TDV5 1/20 0.31
FHIT P49789 1/20 0.30
BACE1 P56817 1/20 0.30
PDE4B Q07343 1/20 0.30
PDE4D Q08499 1/20 0.30
MTNR1B P49286 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8562237 1.00 ESR1 (0.39) ESR1ESR2HDAC6ABHD6LPAR5
SCHEMBL7476930 0.88 DRD2 (0.32)
SCHEMBL7476926 0.88 DRD2 (0.32)
SCHEMBL8564898 0.87 ESR1 (0.39) ESR1ESR2HDAC6ABHD6LPAR5
SCHEMBL8564893 0.87 ESR1 (0.39) ESR1ESR2HDAC6ABHD6LPAR5
SCHEMBL8562570 0.87 DRD2 (0.35) LPAR5
SCHEMBL8562566 0.87 DRD2 (0.35) LPAR5
SCHEMBL8566561 0.85 ESR1 (0.38) ESR1ESR2HDAC6ABHD6BACE1
SCHEMBL8566564 0.85 ESR1 (0.38) ESR1ESR2HDAC6ABHD6BACE1
SCHEMBL7418940 0.83 ESR1 (0.42) ESR1ESR2HDAC6ABHD6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612741-B1 Cyclic derivatives, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1998-06-10 EP disclosed
US-5612335-A ANTICOAGULANTS; COMBATING/PREVENTING DISEASES WHERE CELL AGGREGATES OCCUR OR CELL-MATRIX INTERACTIONS PLAY A PART KARL THOMAE GMBH (DE) 1997-03-18 US disclosed
US-5519036-A IMIDAZOLIDINONES, ANTICOAGULANTS, CELL AGGREGATION PREVENTION KARL THOMAE GMBH (DE) 1996-05-21 US disclosed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP disclosed