SCHEMBL8900813

SCHEMBL8900813

COC(=O)CC(Cl)Cc1ccc(OC)cc1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.56
HTT P42858 1/20 0.47
KMT2A Q03164 1/20 0.47
MMP1 P03956 1/20 0.46
F2RL1 P55085 1/20 0.46
SLC6A4 P31645 1/20 0.46
FPR2 P25090 1/20 0.46
ACACB O00763 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6461540 0.85 LDHA (0.62) LDHAKMT2AMMP1SLC6A4
SCHEMBL8902344 0.82 LDHA (0.57) LDHAHTTMMP1F2RL1SLC6A4
SCHEMBL11837761 0.81 SRR (0.48) HTT
SCHEMBL28062779 0.78 LDHA (0.53) LDHAHTTMMP1F2RL1SLC6A4
SCHEMBL27535459 0.78 LDHA (0.53) LDHAHTTMMP1F2RL1SLC6A4
SCHEMBL11550992 0.77 LDHA (0.56) LDHAHTTF2RL1SLC6A4FPR2
SCHEMBL5672844 0.77 LDHA (0.59) LDHAHTTF2RL1SLC6A4FPR2
SCHEMBL28495195 0.75 LDHA (0.61) LDHAHTTF2RL1SLC6A4FPR2
SCHEMBL7517684 0.75 LDHA (0.71) LDHAHTTKMT2ASLC6A4
SCHEMBL15312744 0.75 LDHA (0.71) LDHAHTTKMT2ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686481-A INDOLE DERIVATIVES; TREATING HYPERTENSION, RENAL FAILURE, CEREBROVASCULAR DISEASE SMITHKLINE BEECHAM CORPORATION (US) 1997-11-11 US disclosed
EP-0676959-A4 ENDOTHELIN RECEPTOR ANTAGONISTS. SMITHKLINE BEECHAM CORP (US) 1996-01-03 EP disclosed
EP-0676959-A1 ENDOTHELIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1995-10-18 EP disclosed
WO-1994014434-A1 ENDOTHELIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1994-07-07 WO disclosed