SCHEMBL8901121

SCHEMBL8901121

COC(C1=CCNCC1)c1ccccc1.OC(C1=CCN(Cc2ccccc2)CC1)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.35
HTR1A P08908 4/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
HTR2A P28223 2/20 0.34
SLC6A4 P31645 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
HTT P42858 1/20 0.34
DRD4 P21917 1/20 0.33
DRD3 P35462 1/20 0.33
ATM Q13315 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8441289 0.81 KDM4E (0.50) DRD2HTR1AKDM4EMEN1KMT2A
SCHEMBL8443999 0.77 SIGMAR1 (0.43) KDM4EMEN1KMT2AHTR2ASIGMAR1
SCHEMBL9387302 0.70 SIGMAR1 (0.46) DRD2HTR1AKDM4EMEN1KMT2A
SCHEMBL8444407 0.69 TACR1 (0.48) DRD2HTR1AKDM4EMEN1KMT2A
SCHEMBL5230745 0.68 KDM4E (0.46) DRD2HTR1AKDM4EMEN1KMT2A
SCHEMBL7948775 0.67 SIGMAR1 (0.48) DRD2HTR1AKDM4EMEN1KMT2A
SCHEMBL28895871 0.66 HDAC4 (0.54) DRD2HTR1AKDM4EMEN1KMT2A
SCHEMBL8441977 0.66 SIGMAR1 (0.42) KDM4EHTR2ASLC6A4SIGMAR1HTT
SCHEMBL10616944 0.66 APOBEC3A (0.48) DRD2HTR1AKDM4EMEN1KMT2A
SCHEMBL28895926 0.66 TACR1 (0.44) DRD2HTR1AKDM4EHTR2ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997017337-A1 SUBSTITUTED 1-INDOLYLPROPYL-4-BENZYL-TETRAHYDROPYRIDINE DERIVATIVES MERCK SHARP & DOHME LIMITED (GB) 1997-05-15 WO disclosed