SCHEMBL8901138

SCHEMBL8901138

O=[N+]([O-])c1cc(Cc2c[c]ccc2)ccc1Cl

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 12/20 0.46
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
POLB P06746 1/20 0.42
KDM1A O60341 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
MEN1 O00255 1/20 0.40
HPGD P15428 1/20 0.40
KMT2A Q03164 1/20 0.40
AKR1B10 O60218 1/20 0.40
AKR1B1 P15121 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9511525 0.82 VCAM1 (0.56) VCAM1ALDH1A1KDM4EPOLBKDM1A
SCHEMBL29936572 0.82 VCAM1 (0.56) VCAM1ALDH1A1KDM4EPOLBKDM1A
SCHEMBL13239653 0.75 VCAM1 (0.50) VCAM1ALDH1A1KDM4EPOLBSMN1; SMN2
SCHEMBL15380348 0.73 VCAM1 (0.54) VCAM1ALDH1A1KDM4EPOLBKDM1A
SCHEMBL28555521 0.73 SMN1; SMN2 (0.59) VCAM1ALDH1A1KDM4EPOLBKDM1A
SCHEMBL4520586 0.72 VCAM1 (0.53) VCAM1ALDH1A1KDM4EPOLBKDM1A
Hydrochloric Acid SCHEMBL29159241 0.72 VCAM1 (0.53) VCAM1ALDH1A1KDM4EPOLBKDM1A
SCHEMBL10389338 0.71 VCAM1 (0.56) VCAM1ALDH1A1KDM4EPOLB
SCHEMBL15600303 0.71 KDM1A (0.54) VCAM1ALDH1A1KDM4EPOLBKDM1A
SCHEMBL2585956 0.71 CALM1 (0.43) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5684205-A CHLORIDE CHANNEL BLOCKERS FOR CONTROLLING AIRWAY DISEASES, SECRETORY DIARRHEA AND ANTIINFLAMMATORY AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1997-11-04 US claimed
EP-0701988-A1 Substituted cyclopentane-di- and triones, their preparation and their use as chloride channel blockers BAYER AG (DE) 1996-03-20 EP claimed
US-5684205-A CHLORIDE CHANNEL BLOCKERS FOR CONTROLLING AIRWAY DISEASES, SECRETORY DIARRHEA AND ANTIINFLAMMATORY AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1997-11-04 US disclosed
EP-0701988-A1 Substituted cyclopentane-di- and triones, their preparation and their use as chloride channel blockers BAYER AG (DE) 1996-03-20 EP disclosed