SCHEMBL8901160

SCHEMBL8901160

CC(C)c1nc2c(c(-c3ccc(F)cc3)c1C#COC(=O)CC(O)C[PH](=O)O)CCCC2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
MAPT P10636 1/20 0.37
KDM4E B2RXH2 3/20 0.36
CACNB4 O00305 2/20 0.36
CACNA1A O00555 2/20 0.36
CACNA1G O43497 2/20 0.36
CACNG3 O60359 2/20 0.36
CACNA1F O60840 2/20 0.36
CACNA1H O95180 2/20 0.36
ACHE P22303 2/20 0.36
CACNB3 P54284 2/20 0.36
CACNA2D1 P54289 2/20 0.36
CACNG7 P62955 2/20 0.36
CACNA1B Q00975 2/20 0.36
CACNA1D Q01668 2/20 0.36
CACNB1 Q02641 2/20 0.36
CACNG1 Q06432 2/20 0.36
CACNB2 Q08289 2/20 0.36
CACNA1S Q13698 2/20 0.36
CACNA1C Q13936 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10345240 0.84 HMGCR (0.39) ALDH1A1MAPTKDM4ECACNB4CACNA1A
SCHEMBL8877671 0.82
SCHEMBL8877479 0.82
SCHEMBL8877485 0.80
SCHEMBL8879918 0.80 HMGCR (0.37)
SCHEMBL8877703 0.77 KDM4E (0.44) MAPTKDM4EADORA2AHPGD
SCHEMBL8877364 0.77 HMGCR (0.43) MAPTKDM4EADORA2AHPGD
SCHEMBL8877344 0.77 KDM4E (0.42) ALDH1A1KDM4EHPGD
SCHEMBL8876404 0.75
SCHEMBL8901153 0.75 KDM4E (0.38) ALDH1A1MAPTKDM4ECACNB4CACNA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686433-A CHOLESTEROL BIOSYNTHESIS INHIBITION E.R. SQUIBB & SONS, INC. (US) 1997-11-11 US disclosed