SCHEMBL10345240

SCHEMBL10345240

CC(C)c1nc2c(c(-c3ccc(F)cc3)c1C#CO[PH](=O)C[C@@H](O)CC(=O)O)CCCC2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 3/20 0.39
ESR1 P03372 1/20 0.39
CHRM1 P11229 1/20 0.39
TBXA2R P21731 1/20 0.39
PDE4A P27815 1/20 0.39
ADRA1A P35348 1/20 0.39
KDM4E B2RXH2 3/20 0.37
CACNB4 O00305 2/20 0.37
CACNA1A O00555 2/20 0.37
CACNA1G O43497 2/20 0.37
CACNG3 O60359 2/20 0.37
CACNA1F O60840 2/20 0.37
CACNA1H O95180 2/20 0.37
ACHE P22303 2/20 0.37
CACNB3 P54284 2/20 0.37
CACNA2D1 P54289 2/20 0.37
CACNG7 P62955 2/20 0.37
CACNA1B Q00975 2/20 0.37
CACNA1D Q01668 2/20 0.37
CACNB1 Q02641 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8901160 0.84 ALDH1A1 (0.37) KDM4ECACNB4CACNA1ACACNA1GCACNG3
SCHEMBL10345388 0.83 SQOR (0.37) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL10345348 0.82 NR4A2 (0.42) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL8953266 0.81
SCHEMBL8953273 0.81
SCHEMBL10345393 0.76
SCHEMBL8901153 0.75 KDM4E (0.38) KDM4ECACNB4CACNA1ACACNA1GCACNG3
SCHEMBL10345400 0.74 CTSA (0.34) HMGCR
SCHEMBL10442264 0.73 HMGCR (0.51) HMGCRALDH1A1
SCHEMBL8877867 0.72 KDM4E (0.39) KDM4ECACNB4CACNA1ACACNA1GCACNG3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0356788-A2 Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1990-03-07 EP claimed
EP-0356788-A2 Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1990-03-07 EP disclosed