SCHEMBL8901408

SCHEMBL8901408

O=C(c1ccccc1)N1CCC(Br)C1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.60
EPHX1 P07099 1/20 0.55
L3MBTL3 Q96JM7 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
HPGD P15428 1/20 0.53
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
ATM Q13315 1/20 0.52
KMT2A Q03164 3/20 0.51
KDM4E B2RXH2 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
SLC18A3 Q16572 1/20 0.51
MEN1 O00255 2/20 0.50
MGLL Q99685 1/20 0.50
SIGMAR1 Q99720 1/20 0.50
HSD11B1 P28845 1/20 0.50
CHRNB2 P17787 1/20 0.50
CHRNB4 P30926 1/20 0.50
CHRNA3 P32297 1/20 0.50
CHRNA7 P36544 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6580374 0.89 ACHE (0.69) ACHEEPHX1L3MBTL3L3MBTL1HPGD
SCHEMBL2720515 0.81 ACHE (0.62) ACHEEPHX1L3MBTL3L3MBTL1HPGD
SCHEMBL4392851 0.81 ACHE (0.62) ACHEEPHX1L3MBTL3L3MBTL1HPGD
SCHEMBL12442621 0.81 ACHE (0.62) ACHEEPHX1L3MBTL3L3MBTL1HPGD
SCHEMBL5871923 0.81 ACHE (0.62) ACHEEPHX1L3MBTL3L3MBTL1HPGD
SCHEMBL2997818 0.79 ACHE (0.60) ACHEEPHX1L3MBTL3L3MBTL1HPGD
SCHEMBL8919161 0.79 SLC18A3 (0.62) ACHEEPHX1L3MBTL3L3MBTL1HPGD
SCHEMBL2130912 0.79 ACHE (0.60) ACHEEPHX1L3MBTL3L3MBTL1HPGD
SCHEMBL18166097 0.79 ACHE (0.81) ACHEEPHX1L3MBTL3L3MBTL1HPGD
SCHEMBL433828 0.79 ACHE (0.81) ACHEEPHX1L3MBTL3L3MBTL1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1042539-C 11,21-bisphenyl-19-norpregnane derivatives AKZO NOBEL NV (NL) 1999-03-17 CN disclosed
EP-0683172-B1 11,21-Bisphenyl-19-norpregnane derivatives AKZO NOBEL NV (NL) 1997-08-13 EP disclosed
US-5620966-A ANTIGLUOCORTICOID ACTIVITY AKZO NOBEL N.V. (NL) 1997-04-15 US disclosed
EP-0683172-A1 11,21-Bisphenyl-19-norpregnane derivatives Akzo Nobel N.V. (NL) 1995-11-22 EP disclosed