SCHEMBL8901822

SCHEMBL8901822

COc1nc(-c2cc(C(C)(C)C)c(O)c(C(C)(C)C)c2)nc2nc[nH]c12

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.46
CTSS P25774 2/20 0.43
CTSK P43235 2/20 0.43
ADORA3 P0DMS8 5/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
PDPK1 O15530 1/20 0.41
ADORA1 P30542 4/20 0.39
PTGS1 P23219 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8902364 0.86 CDK1 (0.52) PTGS2CTSSCTSKPTGS1
SCHEMBL8903318 0.85 CDK1 (0.53) PTGS2CTSSCTSKADORA3ADORA1
SCHEMBL8902849 0.84 CA1 (0.43) PTGS2CTSSCTSKADORA3CA1
SCHEMBL8902911 0.83 CDK1 (0.55) PTGS2CTSSCTSKADORA3PTGS1
SCHEMBL8901655 0.83 CDK1 (0.55) PTGS2CTSSCTSKADORA3PTGS1
SCHEMBL8903387 0.81 CDK1 (0.39) PTGS2CTSSCTSKADORA3
SCHEMBL8902502 0.81 CDK1 (0.55) CTSSCTSKADORA3ADORA1
SCHEMBL8901819 0.80 PTGS2 (0.46) PTGS2CA1CA2PTGS1
SCHEMBL8903452 0.80 CDK1 (0.41) PTGS2CTSSCTSKADORA3
SCHEMBL8903186 0.80 CDK1 (0.41) PTGS2CTSSCTSKADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5602140-A CAUSED BY LEUKOCYTES JAPAN ENERGY CORPORATION (JP) 1997-02-11 US disclosed
EP-0675124-A2 Purine derivatives and suppressants for inflammatory diseases JAPAN ENERGY CORPORATION (JP) 1995-10-04 EP disclosed