SCHEMBL8902502

SCHEMBL8902502

CC(C)(C)c1cc(-c2nc(OCCc3ccccc3)c3[nH]cnc3n2)cc(C(C)(C)C)c1O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 5/20 0.55
CCNB1 P14635 5/20 0.55
CCNA2 P20248 5/20 0.55
CDK2 P24941 5/20 0.55
CCNA1 P78396 5/20 0.55
MGMT P16455 5/20 0.42
PIN1 Q13526 5/20 0.42
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
LMNA P02545 1/20 0.42
TSHR P16473 1/20 0.42
NFKB1 P19838 1/20 0.42
BLM P54132 1/20 0.42
PMP22 Q01453 1/20 0.42
ADORA3 P0DMS8 4/20 0.39
ADORA1 P30542 4/20 0.39
ADORA2A P29274 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8902364 0.85 CDK1 (0.52) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL8903318 0.84 CDK1 (0.53) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL8902498 0.84 CDK1 (0.38) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL8903387 0.83 CDK1 (0.39) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL8901655 0.82 CDK1 (0.55) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL8902911 0.82 CDK1 (0.55) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL8903186 0.81 CDK1 (0.41) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL8901822 0.81 PTGS2 (0.46) ADORA3ADORA1CTSSCTSK
SCHEMBL8903379 0.80 PIN1 (0.43) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL8902849 0.75 CA1 (0.43) ADORA3ADORA1ADORA2ACTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5602140-A CAUSED BY LEUKOCYTES JAPAN ENERGY CORPORATION (JP) 1997-02-11 US claimed
US-5602140-A CAUSED BY LEUKOCYTES JAPAN ENERGY CORPORATION (JP) 1997-02-11 US disclosed
EP-0675124-A2 Purine derivatives and suppressants for inflammatory diseases JAPAN ENERGY CORPORATION (JP) 1995-10-04 EP disclosed