SCHEMBL8904841

SCHEMBL8904841

C[C@H](Oc1ccc(F)cc1[N+](=O)[O-])[C@@H](NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HTT P42858 1/20 0.40
PYGL P06737 2/20 0.38
PDK1 Q15118 1/20 0.38
MAPT P10636 4/20 0.38
TRPA1 O75762 1/20 0.37
PPARG P37231 1/20 0.37
PPARA Q07869 1/20 0.37
AAK1 Q2M2I8 1/20 0.36
CTSS P25774 2/20 0.36
CTSK P43235 2/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1561567 1.00 ALDH1A1 (0.40) ALDH1A1L3MBTL1HTTPYGLPDK1
SCHEMBL8904838 1.00 ALDH1A1 (0.40) ALDH1A1L3MBTL1HTTPYGLPDK1
SCHEMBL27391920 1.00 ALDH1A1 (0.40) ALDH1A1L3MBTL1HTTPYGLPDK1
SCHEMBL8904801 0.92 ALDH1A1 (0.46) ALDH1A1L3MBTL1HTTPYGLMAPT
SCHEMBL8904797 0.92 ALDH1A1 (0.46) ALDH1A1L3MBTL1HTTPYGLMAPT
SCHEMBL27372381 0.92 ALDH1A1 (0.46) ALDH1A1L3MBTL1HTTPYGLMAPT
SCHEMBL1561729 0.88 MAPT (0.53) ALDH1A1L3MBTL1HTTMAPTPPARG
SCHEMBL29079146 0.88 AAK1 (0.43) ALDH1A1PDK1MAPTPPARGPPARA
SCHEMBL1562131 0.87 ALDH1A1 (0.43) ALDH1A1HTTMAPTPPARGPPARA
SCHEMBL9221220 0.87 ALDH1A1 (0.43) ALDH1A1HTTMAPTPPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5618808-A Benzothiazepine and benzoxazepine derivatives as cholecystokinin receptor antagonists PFIZER, INC. (US) 1997-04-08 US disclosed
EP-0648213-A1 BENZOTHIAZEPINE AND BENZOXAZEPINE DERIVATIVES AS CHOLECYSTOKININ RECEPTOR ANTAGONISTS PFIZER INC. (US) 1995-04-19 EP disclosed
WO-1994001421-A1 BENZOTHIAZEPINE AND BENZOXAZEPINE DERIVATIVES AS CHOLECYSTOKININ RECEPTOR ANTAGONISTS PFIZER INC. (US) 1994-01-20 WO disclosed