SCHEMBL8905142

SCHEMBL8905142

COc1cccc(NC(=O)NC2CSc3ccccc3N(CC(=O)N3CCCCC3C)C2=O)c1

nearest known ligand 0.61

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 12/20 0.61
ALDH1A1 P00352 3/20 0.46
MAPT P10636 3/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
HTT P42858 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
NPY1R P25929 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8905144 1.00 CCKBR (0.61) CCKBRALDH1A1MAPTMEN1KMT2A
SCHEMBL8905133 0.90 CCKBR (0.59) CCKBRALDH1A1MAPTMEN1KMT2A
SCHEMBL8905125 0.90 CCKBR (0.59) CCKBRALDH1A1MAPTMEN1KMT2A
SCHEMBL8904898 0.84 CCKBR (0.63) CCKBRALDH1A1MAPTMEN1KMT2A
SCHEMBL8904459 0.83 CCKBR (0.62) CCKBRALDH1A1MAPTMEN1KMT2A
SCHEMBL8905718 0.83 CCKBR (0.62) CCKBRALDH1A1MAPTMEN1KMT2A
SCHEMBL8904134 0.83 CCKBR (0.62) CCKBRALDH1A1MAPTMEN1KMT2A
SCHEMBL8903044 0.83 CCKBR (0.62) CCKBRALDH1A1MAPTMEN1KMT2A
SCHEMBL8903048 0.83 CCKBR (0.62) CCKBRALDH1A1MAPTMEN1KMT2A
SCHEMBL8905490 0.81 CCKBR (0.54) CCKBRALDH1A1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5618808-A Benzothiazepine and benzoxazepine derivatives as cholecystokinin receptor antagonists PFIZER, INC. (US) 1997-04-08 US disclosed