SCHEMBL8905217

SCHEMBL8905217

CCCc1nc2cc(-c3nc4ccccc4n3C)ccc2n1-c1cccc(-c2ccccc2-c2nnn[nH]2)c1C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.37
ALDH1A1 P00352 4/20 0.37
HSD17B10 Q99714 3/20 0.37
PPARG P37231 2/20 0.37
ABCC3 O15438 1/20 0.37
ABCC4 O15439 1/20 0.37
USP2 O75604 1/20 0.37
ABCB11 O95342 1/20 0.37
CHRM2 P08172 1/20 0.37
CYP3A4 P08684 1/20 0.37
ADRA2A P08913 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
CHRM1 P11229 1/20 0.37
CYP2C9 P11712 1/20 0.37
ACE P12821 1/20 0.37
ADRA2C P18825 1/20 0.37
TBXA2R P21731 1/20 0.37
GLRA1 P23415 1/20 0.37
PDE4A P27815 1/20 0.37
HTR2A P28223 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8905808 0.95 ALDH1A1 (0.39) KDM4EALDH1A1HSD17B10PPARGABCC3
SCHEMBL8907620 0.90 AGTR1 (0.38) KDM4EALDH1A1HSD17B10PPARGABCC3
SCHEMBL8905630 0.89 KDM4E (0.39) KDM4EALDH1A1HSD17B10PPARGABCC3
SCHEMBL8905214 0.86 PPARG (0.37) KDM4EALDH1A1HSD17B10PPARGABCC3
SCHEMBL8905654 0.83 PPARG (0.31) PPARGAGTR1AGTR2
SCHEMBL8906823 0.83 ALDH1A1 (0.41) KDM4EALDH1A1HSD17B10BRD4NPC1
SCHEMBL8907540 0.82 CYP3A4 (0.31) PPARGCYP3A4AGTR1AGTR2
SCHEMBL8789663 0.81 PPARG (0.53) KDM4EALDH1A1HSD17B10PPARGABCC3
SCHEMBL8905695 0.81 PPARG (0.54) KDM4EALDH1A1HSD17B10PPARGABCC3
SCHEMBL8905804 0.81 KDM4E (0.40) KDM4EALDH1A1HSD17B10PPARGABCC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5684029-A HYPOTENSIVE AGENTS KARL THOMAE GMBH (DE) 1997-11-04 US disclosed