SCHEMBL8905546

SCHEMBL8905546

CCCCc1nc2ccc(-c3nccn3CCCC)cc2n1-c1ccc(-c2ccccc2)c(-c2nnn[nH]2)c1C

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.34
CYP2C19 P33261 2/20 0.34
TSHR P16473 1/20 0.34
AGTR1 P30556 2/20 0.34
AGTR2 P50052 2/20 0.34
CYP2C9 P11712 1/20 0.34
HIF1A Q16665 1/20 0.34
PDE6D O43924 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8905653 0.94 CYP3A4 (0.35) CYP3A4CYP2C19TSHRAGTR1AGTR2
SCHEMBL8907533 0.93 CYP3A4 (0.34) CYP3A4CYP2C19TSHRAGTR1CYP2C9
SCHEMBL8905755 0.93 AGTR1 (0.33) AGTR1AGTR2
SCHEMBL8905647 0.88 CYP1A2 (0.33)
SCHEMBL8907613 0.88 AGTR1 (0.37) CYP3A4AGTR1AGTR2CYP2C9
SCHEMBL8905553 0.87 AGTR1 (0.33) CYP3A4CYP2C19TSHRAGTR1AGTR2
SCHEMBL8906964 0.83 AGTR1 (0.31) AGTR1AGTR2
SCHEMBL8906938 0.83 AGTR1 (0.32) AGTR1AGTR2
SCHEMBL8907815 0.83 CYP1A2 (0.32)
SCHEMBL8905804 0.83 KDM4E (0.40) CYP3A4AGTR1AGTR2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5684029-A HYPOTENSIVE AGENTS KARL THOMAE GMBH (DE) 1997-11-04 US disclosed