SCHEMBL8905660

SCHEMBL8905660

CCCCCCn1ccnc1-c1ccc2nc(CCC)n(-c3cccc(-c4ccccc4-c4nnn[nH]4)c3C)c2c1

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.33
CYP2C19 P33261 2/20 0.33
TSHR P16473 1/20 0.33
TP53 P04637 1/20 0.31
CYP2C9 P11712 1/20 0.31
HIF1A Q16665 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8905553 0.94 AGTR1 (0.33) CYP3A4CYP2C19TSHRCYP2C9HIF1A
SCHEMBL8907540 0.94 CYP3A4 (0.31) CYP3A4CYP2C19TSHR
SCHEMBL8905654 0.90 PPARG (0.31)
SCHEMBL8905761 0.88 AGTR1 (0.33)
SCHEMBL8905653 0.88 CYP3A4 (0.35) CYP3A4CYP2C19TSHRTP53CYP2C9
SCHEMBL8907819 0.85 PIK3R2 (0.31)
SCHEMBL8906071 0.84 PIK3R2 (0.30)
SCHEMBL8905808 0.84 ALDH1A1 (0.39) CYP3A4TP53CYP2C9
SCHEMBL8791417 0.83 AGTR1 (0.45)
SCHEMBL8905754 0.83 PPARG (0.44) CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5684029-A HYPOTENSIVE AGENTS KARL THOMAE GMBH (DE) 1997-11-04 US disclosed