SCHEMBL8906158

SCHEMBL8906158

Cn1c(Cc2ccc(=O)[nH]n2)ccc1C(=O)c1ccc(Cl)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
POLB P06746 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP3A4 P08684 2/20 0.40
CYP2C19 P33261 2/20 0.39
CYP1A2 P05177 1/20 0.39
AKR1B1 P15121 2/20 0.38
THRA P10827 1/20 0.38
RAB9A P51151 2/20 0.37
MAPT P10636 1/20 0.37
SRD5A2 P31213 1/20 0.36
P2RX7 Q99572 1/20 0.36
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 2/20 0.35
LMNA P02545 2/20 0.35
GLA P06280 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9030680 0.87 CYP3A4 (0.37) SMN1; SMN2KMT2APOLBCYP2C9CYP3A4
SCHEMBL8905896 0.84 PTGS2 (0.41) SMN1; SMN2CYP3A4CYP1A2AKR1B1ALDH1A1
SCHEMBL8905529 0.83 CYP3A4 (0.53) CYP3A4AKR1B1RAB9ANPC1ALDH1A1
SCHEMBL8904324 0.82 AKR1B1 (0.39) MEN1KMT2ACYP3A4AKR1B1RAB9A
SCHEMBL8904844 0.78 AKR1B1 (0.43) SMN1; SMN2HSD17B10MEN1KMT2ACYP3A4
SCHEMBL9030256 0.77 CXCL8 (0.40) MEN1KMT2ACYP3A4AKR1B1RAB9A
SCHEMBL8905800 0.77 AKR1B1 (0.54) SMN1; SMN2MEN1KMT2APOLBCYP2C9
SCHEMBL8904081 0.76 CXCL8 (0.40) SMN1; SMN2MEN1KMT2APOLBCYP3A4
SCHEMBL9031112 0.76 CXCL8 (0.40) SMN1; SMN2MEN1KMT2APOLBCYP3A4
SCHEMBL8904190 0.76 AKR1B1 (0.41) SMN1; SMN2MEN1KMT2ACYP3A4AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5622948-A ANALGESICS SYNTEX (U.S.A.) INC. (US) 1997-04-22 US disclosed
EP-0714895-A1 Pyrrole derivatives F. Hoffmann-La Roche AG (CH) 1996-06-05 EP disclosed