SCHEMBL8907669

SCHEMBL8907669

OCCC#Cc1cnc2ccccc2c1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.77
ACACB O00763 1/20 0.45
CYP1A2 P05177 1/20 0.42
PDGFRB P09619 3/20 0.41
PDGFRA P16234 3/20 0.41
MGAM O43451 1/20 0.41
RAB9A P51151 2/20 0.40
ASIC3 Q9UHC3 1/20 0.40
BIRC5 O15392 1/20 0.39
TLR8 Q9NR97 1/20 0.38
EGFR P00533 1/20 0.38
PIK3CA P42336 2/20 0.38
PIK3CD O00329 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MTOR P42345 1/20 0.38
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3059701 0.90 ALDH1A1 (0.71) ALDH1A1ACACBCYP1A2PDGFRBPDGFRA
SCHEMBL372200 0.87 ALDH1A1 (1.00) ALDH1A1ACACBCYP1A2PDGFRBPDGFRA
SCHEMBL12603967 0.82 ALDH1A1 (0.64) ALDH1A1ACACBCYP1A2RAB9ATLR8
SCHEMBL13356421 0.82 ALDH1A1 (0.64) ALDH1A1ACACBCYP1A2PDGFRBPDGFRA
SCHEMBL23781564 0.81 ALDH1A1 (0.71) ALDH1A1ACACBCYP1A2PDGFRBPDGFRA
SCHEMBL10162702 0.81 ALDH1A1 (0.71) ALDH1A1ACACBCYP1A2PDGFRBPDGFRA
SCHEMBL12603955 0.79 ALDH1A1 (0.64) ALDH1A1ACACBCYP1A2PDGFRBPDGFRA
SCHEMBL10130641 0.77 ALDH1A1 (0.66) ALDH1A1ACACBCYP1A2PDGFRBPDGFRA
SCHEMBL6881031 0.77 ALDH1A1 (0.66) ALDH1A1ACACBCYP1A2PDGFRBPDGFRA
SCHEMBL6847857 0.77 ALDH1A1 (0.65) ALDH1A1ACACBCYP1A2PDGFRBPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5620988-A Substituted tetrahydropyridines and hydroxypiperidines as central nervous system agents WARNER-LAMBERT COMPANY (US) 1997-04-15 US disclosed
EP-0556332-B1 SUBSTITUTED TETRAHYDROPYRIDINES AND HYDROXYPIPERIDINES AS CENTRAL NERVOUS SYSTEM AGENTS WARNER LAMBERT CO (US) 1996-03-20 EP disclosed
EP-0556329-B1 SUBSTITUTED PIPERAZINES AS CENTRAL NERVOUS SYSTEM AGENTS WARNER LAMBERT CO (US) 1996-01-10 EP disclosed
US-5466698-A Substituted tetrahydrophyridines and hydroxypiperidines as central nervous system agents WARNER-LAMBERT COMPANY (US) 1995-11-14 US disclosed
US-5273977-A 1-Phenylethylidynealkylene-4-phenyl-1,2,5,6-tetrahydropyridines WARNER-LAMBERT COMPANY (US) 1993-12-28 US disclosed
US-5270312-A Substituted piperazines as central nervous system agents WARNER-LAMBERT COMPANY (US) 1993-12-14 US disclosed
US-5187280-A Dopaminergic, antipsychotic and antihypertensive agents WARNER-LAMBERT COMPANY (US) 1993-02-16 US disclosed
US-5118691-A Substituted tetrahydropyridines as central nervous system agents WARNER-LAMBERT CO. (US) 1992-06-02 US disclosed
WO-1992007831-A1 SUBSTITUTED TETRAHYDROPYRIDINES AND HYDROXYPIPERIDINES AS CENTRAL NERVOUS SYSTEM AGENTS WARNER-LAMBERT COMPANY (US) 1992-05-14 WO disclosed
US-5045550-A Antipsychotic, hypotensive agents, dopaminergic WARNER-LAMBERT CO. (US) 1991-09-03 US disclosed