SCHEMBL8907692

SCHEMBL8907692

CCCc1cc(C(=O)OC)ccc1C=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 6/20 0.48
ALDH1A1 P00352 6/20 0.47
PPARG P37231 3/20 0.46
PPARA Q07869 3/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
ATM Q13315 1/20 0.46
HCRTR1 O43613 1/20 0.45
HCRTR2 O43614 1/20 0.45
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
XDH P47989 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
ALOX15 P16050 1/20 0.42
HTT P42858 1/20 0.42
KDM4E B2RXH2 4/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8907608 0.87 PPARG (0.45) ALDH1A1PPARGPPARAL3MBTL1KMT2A
SCHEMBL28329861 0.83 ERN1 (0.49) ERN1ALDH1A1ATMHCRTR1HCRTR2
SCHEMBL10020273 0.83 ERN1 (0.49) ERN1ALDH1A1ATMHCRTR1HCRTR2
SCHEMBL12419937 0.81 PPARG (0.50) ALDH1A1PPARGPPARAL3MBTL1KMT2A
SCHEMBL15337170 0.80 PPARG (0.51) ALDH1A1PPARGPPARAL3MBTL1KMT2A
SCHEMBL542559 0.80 CA1 (0.61) ALDH1A1PPARGPPARAL3MBTL1KMT2A
SCHEMBL30232935 0.80 CA1 (0.61) ALDH1A1PPARGPPARAL3MBTL1KMT2A
SCHEMBL17747083 0.79 ALDH1A1 (0.58) ERN1ALDH1A1KMT2AMEN1ATM
SCHEMBL8906623 0.78 PPARG (0.48) ALDH1A1PPARGPPARAL3MBTL1KMT2A
SCHEMBL3273922 0.78 CCR6 (0.49) ALDH1A1PPARGPPARAL3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686478-A Endothelin antagonists MERCK & CO. INC. (US) 1997-11-11 US disclosed
EP-0710235-A4 1996-06-12 EP disclosed
EP-0710235-A1 ENDOTHELIN ANTAGONISTS MERCK & CO. INC. (US) 1996-05-08 EP disclosed
WO-1995003295-A1 ENDOTHELIN ANTAGONISTS MERCK & CO., INC. (US) 1995-02-02 WO disclosed