SCHEMBL8907855

SCHEMBL8907855

CCC(O)Nc1ccc(F)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.46
MMP2 P08253 1/20 0.46
ALDH1A1 P00352 3/20 0.45
TDP1 Q9NUW8 3/20 0.45
THRB P10828 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
TP53 P04637 1/20 0.45
HSP90AA1 P07900 1/20 0.45
CYP3A4 P08684 1/20 0.45
ALOX15 P16050 1/20 0.45
TSHR P16473 1/20 0.45
CASP1 P29466 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HIF1A Q16665 1/20 0.45
HSD17B10 Q99714 1/20 0.45
KCNH3 Q9ULD8 1/20 0.40
CXCL12 P48061 1/20 0.40
MAPT P10636 4/20 0.40
KDM4E B2RXH2 4/20 0.40
MEN1 O00255 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL447463 0.81 CA12 (0.47) CA12ALDH1A1TDP1THRBL3MBTL1
SCHEMBL14532077 0.79 CYP3A4 (0.45) ALDH1A1TDP1THRBL3MBTL1TP53
SCHEMBL445994 0.79 TDP1 (0.45) CA12ALDH1A1TDP1THRBL3MBTL1
SCHEMBL31265919 0.79 ALDH1A1 (0.75) CA12ALDH1A1TDP1THRBL3MBTL1
SCHEMBL347685 0.78 TDP1 (0.50) CA12ALDH1A1TDP1THRBL3MBTL1
SCHEMBL3088720 0.78 TDP1 (0.48) CA12MMP2ALDH1A1TDP1THRB
SCHEMBL26419568 0.77 CA12 (0.51) CA12MMP2ALDH1A1L3MBTL1TSHR
Hydrochloric Acid SCHEMBL29730240 0.77 TDP1 (0.48) CA12ALDH1A1TDP1THRBL3MBTL1
SCHEMBL27928253 0.77 TDP1 (0.48) CA12ALDH1A1TDP1THRBL3MBTL1
Ammonia Solution, Strong SCHEMBL27928251 0.77 TDP1 (0.48) CA12ALDH1A1TDP1THRBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1249233-B9 NPYY5 ANTAGONISTS SHIONOGI & CO (JP) 2009-08-05 EP disclosed
EP-1249233-B1 NPYY5 ANTAGONISTS SHIONOGI & CO (JP) 2008-08-20 EP disclosed
US-5672605-A ADMINISTERING TO TREAT AUTOIMMUNE DISORDERS, TRANSPLANT REJECTION ABBOTT LABORATORIES (US) 1997-09-30 US disclosed
US-5583139-A Marcolide immunomodulators ABBOTT LABORATORIES (US) 1996-12-10 US disclosed
WO-1995014023-A1 SEMISYNTHETIC ANALOGS OF RAPAMYCIN (MACROLIDES) BEING IMMUNOMODULATORS ABBOTT LABORATORIES (US) 1995-05-26 WO disclosed