Tetraxetan

Tetraxetan

SCHEMBL8907977

O=C(O)CN1CCN(CC(=O)O)CCN(CC(=O)O)CCN(CC(=O)O)CC1.S=C=Nc1ccc(CCN2CCNCCNCCNCC2)cc1

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.48
TP53 P04637 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
ALOX12 P18054 1/20 0.48
KCNH2 Q12809 4/20 0.43
KCNJ1 P48048 2/20 0.43
P2RY6 Q15077 1/20 0.42
GRIN1 Q05586 1/20 0.41
GRIN2A Q12879 1/20 0.41
GRIN2B Q13224 1/20 0.41
SIGMAR1 Q99720 3/20 0.40
SLC6A4 P31645 2/20 0.39
HSD17B10 Q99714 1/20 0.38
TSHR P16473 1/20 0.38
CYP2C19 P33261 1/20 0.38
HIF1A Q16665 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A3 Q01959 1/20 0.38
S1PR1 P21453 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14312096 0.99 CYP2D6 (0.49) CYP2D6TP53CYP1A2CYP3A4ALOX12
SCHEMBL14312072 0.94 CYP2D6 (0.46) CYP2D6TP53CYP1A2CYP3A4ALOX12
SCHEMBL14327160 0.94 CYP2D6 (0.50) CYP2D6TP53CYP1A2CYP3A4ALOX12
SCHEMBL14478355 0.92 CYP2D6 (0.46) CYP2D6TP53CYP1A2CYP3A4ALOX12
SCHEMBL8654441 0.92 CYP2D6 (0.54) CYP2D6TP53CYP1A2CYP3A4ALOX12
SCHEMBL14477644 0.89 CYP2D6 (0.42) CYP2D6TP53CYP1A2CYP3A4ALOX12
SCHEMBL9122681 0.88 P2RY6 (0.54) CYP2D6TP53CYP1A2CYP3A4ALOX12
SCHEMBL14327153 0.87 CYP2D6 (0.41) CYP2D6TP53CYP1A2CYP3A4ALOX12
SCHEMBL26241122 0.87 CYP2D6 (0.53) CYP2D6TP53CYP1A2CYP3A4ALOX12
SCHEMBL14312212 0.87 SIGMAR1 (0.46) P2RY6GRIN1GRIN2AGRIN2BSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5652361-A ANTITUMOR THE DOW CHEMICAL COMPANY (US) 1997-07-29 US disclosed