SCHEMBL8909101

SCHEMBL8909101

Cc1cc(NC(=O)c2ccccc2O)no1

nearest known ligand 0.76

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 9/20 0.76
NPC1 O15118 7/20 0.76
SMN1; SMN2 Q16637 2/20 0.72
CYP1A2 P05177 1/20 0.72
CYP2C19 P33261 1/20 0.72
MEN1 O00255 2/20 0.66
KMT2A Q03164 2/20 0.66
GAA P10253 3/20 0.64
TSHR P16473 3/20 0.64
ALOX15 P16050 2/20 0.64
MAPK1 P28482 1/20 0.64
ALDH1A1 P00352 3/20 0.61
HPGD P15428 3/20 0.61
PKM P14618 2/20 0.61
KDM4E B2RXH2 4/20 0.60
MAPT P10636 1/20 0.59
HSD17B10 Q99714 2/20 0.58
TDP1 Q9NUW8 1/20 0.58
TP53 P04637 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27792444 0.88 RAB9A (0.68) RAB9ANPC1SMN1; SMN2CYP1A2CYP2C19
SCHEMBL27730037 0.84 RAB9A (0.80) RAB9ANPC1SMN1; SMN2CYP1A2CYP2C19
SCHEMBL27771282 0.84 PKM (0.63) RAB9ANPC1SMN1; SMN2CYP1A2CYP2C19
SCHEMBL30788250 0.80 RAB9A (1.00) RAB9ANPC1SMN1; SMN2CYP1A2CYP2C19
SCHEMBL28551813 0.79 RAB9A (0.67) RAB9ANPC1SMN1; SMN2CYP1A2CYP2C19
SCHEMBL8910219 0.79 RAB9A (0.76) RAB9ANPC1SMN1; SMN2CYP1A2CYP2C19
SCHEMBL13055933 0.78 P2RX1 (0.55) RAB9ANPC1SMN1; SMN2CYP1A2CYP2C19
SCHEMBL16363834 0.78 RAB9A (0.74) RAB9ANPC1SMN1; SMN2CYP1A2CYP2C19
SCHEMBL13116740 0.77 RAB9A (0.69) RAB9ANPC1SMN1; SMN2CYP1A2CYP2C19
SCHEMBL30975216 0.76 RAB9A (0.76) RAB9ANPC1SMN1; SMN2CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5622953-A DRUG RESISTANT TO ANTICANCER CHEMOTHERAPEUTIC DRUG BASF AKTIENGESELLSCHAFT (DE) 1997-04-22 US disclosed
EP-0691962-A1 1-AMINO-3-PHENOXY PROPANE DERIVATIVES AS MODULATORS OF MULTI-DRUG RESISTANCE BASF AKTIENGESELLSCHAFT (DE) 1996-01-17 EP disclosed
WO-1994022842-A1 1-AMINO-3-PHENOXY PROPANE DERIVATIVES AS MODULATORS OF MULTI-DRUG RESISTANCE BASF AKTIENGESELLSCHAFT (DE) 1994-10-13 WO disclosed