SCHEMBL8909274

SCHEMBL8909274

CC1(C)CCC(=O)c2cc(-c3ccc4cc(O)ccc4c3)ccc21

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RARB P10826 4/20 0.45
RARG P13631 4/20 0.45
RARA P10276 3/20 0.45
ESR1 P03372 10/20 0.44
ESR2 Q92731 10/20 0.44
ABL1 P00519 2/20 0.41
ABCB1 P08183 2/20 0.41
BCR P11274 2/20 0.41
HSD17B1 P14061 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2B6 P20813 1/20 0.41
CYP2C19 P33261 1/20 0.41
HSD17B2 P37059 1/20 0.41
PBRM1 Q86U86 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8662092 0.85 PBRM1 (0.53) ESR1ESR2HSD17B1CYP3A4PBRM1
SCHEMBL31650524 0.85 PBRM1 (0.53) ESR1ESR2HSD17B1CYP3A4PBRM1
SCHEMBL6423981 0.83 RARB (0.68) RARBRARGRARA
SCHEMBL6419013 0.79 SIRT1 (0.41) RARBRARGRARAESR1ESR2
SCHEMBL10834419 0.78 RARA (0.64) RARBRARGRARAESR1ESR2
SCHEMBL6294335 0.78 RARA (0.48) RARBRARGRARA
Methane SCHEMBL10834484 0.77 RARA (0.62) RARBRARGRARAESR1ESR2
SCHEMBL1806400 0.76 PBRM1 (0.49) ESR1ESR2HSD17B1CYP3A4PBRM1
SCHEMBL8661522 0.75 NSD2 (0.41) RARBRARGRARAESR1ESR2
SCHEMBL445935 0.73 MALT1 (0.41) ESR1ESR2PBRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997048672-A2 SUBSTITUTED TETRAHYDRONAPHTHALENE AND DIHYDRONAPHTHALENE DERIVATIVES HAVING RETINOID AND/OR RETINOID ANTAGONIST-LIKE BIOLOGICAL ACTIVITY ALLERGAN SALES, INC. (US) 1997-12-24 WO disclosed