SCHEMBL8910043

SCHEMBL8910043

O=CC1c2ccccc2COc2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.40
HTR2C P28335 2/20 0.40
HRH1 P35367 2/20 0.40
MAOB P27338 4/20 0.37
MAOA P21397 3/20 0.37
TERT O14746 1/20 0.37
OXTR P30559 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 1/20 0.35
MAPK1 P28482 1/20 0.35
NOTUM Q6P988 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HSD17B3 P37058 1/20 0.34
KMT2A Q03164 1/20 0.33
NPC1 O15118 1/20 0.33
LMNA P02545 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8797201 0.83 KMT2A (0.39) HTR2AHTR2CHRH1TERTGAA
SCHEMBL28428106 0.82 MAOB (0.41) HTR2AHTR2CHRH1MAOBMAOA
SCHEMBL68805 0.77 MAOA (0.52) MAOBMAOAMAPK1KMT2ALMNA
SCHEMBL30138896 0.77 MAOA (0.52) MAOBMAOAMAPK1KMT2ALMNA
SCHEMBL11525800 0.77 HTR2A (0.52) HTR2AHTR2CHRH1MAOA
SCHEMBL2601579 0.77 ACP3 (0.48) HTR2AHTR2C
SCHEMBL8798040 0.76 TBXA2R (0.43) KDM4EALDH1A1GAAHPGDMAPK1
SCHEMBL9185773 0.76 HTR2A (0.43) HTR2AHTR2CHRH1MAOBMAOA
Hydrochloric Acid SCHEMBL28311470 0.75 MAOA (0.50) MAOBMAOAMAPK1KMT2ALMNA
SCHEMBL4465669 0.73 MAOA (0.59) HTR2AHTR2CHRH1MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5622953-A DRUG RESISTANT TO ANTICANCER CHEMOTHERAPEUTIC DRUG BASF AKTIENGESELLSCHAFT (DE) 1997-04-22 US disclosed
EP-0691962-A1 1-AMINO-3-PHENOXY PROPANE DERIVATIVES AS MODULATORS OF MULTI-DRUG RESISTANCE BASF AKTIENGESELLSCHAFT (DE) 1996-01-17 EP disclosed
US-5405843-A Anticancer drug potentiators MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1995-04-11 US disclosed
EP-0363212-B1 Novel heterocyclic compounds and anticancer-drug reinforcing agents containing them as effective components MITSUI TOATSU CHEMICALS (JP) 1995-01-04 EP disclosed
US-5204348-A Quinoline derivatives MITSUI TOATSU CHEMICALS INC. (JP) 1993-04-20 US disclosed
US-5112817-A Anticancer Drug Potentiators MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1992-05-12 US disclosed
EP-0363212-A2 Novel heterocyclic compounds and anticancer-drug reinforcing agents containing them as effective components MITSUI TOATSU CHEMICALS, Inc. (JP) 1990-04-11 EP disclosed