SCHEMBL8910046

SCHEMBL8910046

C[CH][C@H](N)Oc1ccccc1OC(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 2/20 0.46
ALDH1A1 P00352 3/20 0.43
ACHE P22303 1/20 0.43
TLR8 Q9NR97 1/20 0.42
NISCH Q9Y2I1 2/20 0.39
ADRA2A P08913 1/20 0.39
ADRA2B P18089 1/20 0.39
ADRA2C P18825 1/20 0.39
MCHR1 Q99705 1/20 0.39
NPSR1 Q6W5P4 1/20 0.38
CYP1A2 P05177 1/20 0.38
MAPT P10636 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
KDM4E B2RXH2 2/20 0.37
LMNA P02545 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11543855 0.80 SCN4A (0.43) ALDH1A1ACHENISCHADRA2BCYP1A2
SCHEMBL29591819 0.80 ALDH1A1 (0.57) IRAK4ALDH1A1ACHETLR8NISCH
SCHEMBL2069775 0.80 ALDH1A1 (0.57) IRAK4ALDH1A1ACHETLR8NISCH
SCHEMBL7054838 0.75 ALDH1A1 (0.46) IRAK4ALDH1A1ACHETLR8NISCH
SCHEMBL28851801 0.73 ALDH1A1 (0.52) IRAK4ALDH1A1ACHETLR8NISCH
SCHEMBL8909407 0.72 CA4 (0.39) CYP1A2CYP2C9CYP2C19KDM4EPOLB
SCHEMBL366155 0.72 CA4 (0.39) CYP1A2CYP2C9CYP2C19KDM4EPOLB
SCHEMBL31433095 0.72 CA1 (0.65) IRAK4ALDH1A1ACHENISCHADRA2A
SCHEMBL105697 0.72 CA1 (0.65) IRAK4ALDH1A1ACHENISCHADRA2A
SCHEMBL5412728 0.71 ALDH1A1 (0.44) IRAK4ALDH1A1ACHETLR8NISCH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5672588-A Purine derivatives NOVO NORDISK A/S (DK) 1997-09-30 US disclosed
EP-0603348-A1 PURINE DERIVATIVES NOVO NORDISK A/S (DK) 1994-06-29 EP disclosed
WO-1993023418-A1 PURINE DERIVATIVES NOVO NORDISK A/S (DK) 1993-11-25 WO disclosed