SCHEMBL8910129

SCHEMBL8910129

CCC(CC)(CNCc1ccc2sc(-c3ccccc3C#N)cc2c1)C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 2/20 0.38
HDAC1 Q13547 3/20 0.36
PTPN1 P18031 1/20 0.34
CTSB P07858 1/20 0.31
CTSS P25774 1/20 0.31
CTSK P43235 1/20 0.31
S1PR3 Q99500 1/20 0.31
CD274 Q9NZQ7 1/20 0.31
CTSD P07339 1/20 0.31
BACE1 P56817 1/20 0.31
BACE2 Q9Y5Z0 1/20 0.31
HDAC6 Q9UBN7 1/20 0.30
NR1H2 P55055 1/20 0.30
MYC P01106 1/20 0.30
WDR5 P61964 1/20 0.30
RORC P51449 1/20 0.30
NSD2 O96028 1/20 0.30
SLC22A12 Q96S37 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8910135 0.82 PTPN1 (0.32) S1PR1PTPN1S1PR3SLC22A12
SCHEMBL8482788 0.81 PTPN1 (0.34) PTPN1CTSBCTSSCTSKCD274
SCHEMBL8911110 0.79 LTB4R2 (0.34) PTPN1CTSBCTSS
SCHEMBL9079126 0.73 S1PR1 (0.35) S1PR1HDAC1CD274MYCWDR5
SCHEMBL8485600 0.71 MAOB (0.41) CD274HDAC6MYCWDR5
SCHEMBL2200 0.71 MYC (0.45) S1PR1PTPN1S1PR3CD274CTSD
SCHEMBL8484313 0.69 PPARG (0.33) S1PR1HDAC1
SCHEMBL8482925 0.67 ABL1 (0.40) S1PR1PTPN1S1PR3CD274CTSD
SCHEMBL8487337 0.65 CYP2A6 (0.40)
SCHEMBL2226 0.64 MYC (0.46) S1PR1PTPN1S1PR3CD274CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5620998-A CARDIOVASCULAR DISORDERS; HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1997-04-15 US disclosed
US-5506240-A HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1996-04-09 US disclosed