SCHEMBL8910135

SCHEMBL8910135

CCC(CN)(CCCc1ccc2sc(-c3ccccc3C#N)cc2c1)C(=O)OC(C)(C)C

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.32
S1PR1 P21453 1/20 0.32
S1PR3 Q99500 1/20 0.32
SLC22A12 Q96S37 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8910129 0.82 S1PR1 (0.38) PTPN1S1PR1S1PR3SLC22A12
SCHEMBL8482791 0.82 HRH3 (0.34) PTPN1S1PR1S1PR3
SCHEMBL8911110 0.80 LTB4R2 (0.34) PTPN1
SCHEMBL8485604 0.73 MAOB (0.37) S1PR1
SCHEMBL8484313 0.67 PPARG (0.33) S1PR1
SCHEMBL8482788 0.64 PTPN1 (0.34) PTPN1SLC22A12
SCHEMBL8487337 0.64 CYP2A6 (0.40)
SCHEMBL9842996 0.63 AGTR1 (0.51)
SCHEMBL8911282 0.63 LTB4R2 (0.34)
SCHEMBL8482148 0.63 LTB4R2 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5620998-A CARDIOVASCULAR DISORDERS; HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1997-04-15 US disclosed
US-5506240-A HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1996-04-09 US disclosed