SCHEMBL8910139

SCHEMBL8910139

CN1CCc2c(Cl)ccc(CO)c2CC1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 6/20 0.52
ADRA2B P18089 6/20 0.52
ADRA2C P18825 6/20 0.52
ADRA1D P25100 5/20 0.50
ADRA1A P35348 5/20 0.50
ADRA1B P35368 5/20 0.50
CYP2D6 P10635 1/20 0.50
NPSR1 Q6W5P4 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8911862 0.84 ADRA2A (0.48) ADRA2AADRA2BADRA2CADRA1DADRA1A
Hydrochloric Acid SCHEMBL8912304 0.83 ADRA2A (0.47) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL8911419 0.83 ADRA2A (0.52) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL8910076 0.82 ADRA2A (0.46) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL8911196 0.79 ADRA2A (0.52) ADRA2AADRA2BADRA2CADRA1DADRA1A
Hydrochloric Acid SCHEMBL8910878 0.78 ADRA2A (0.51) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL8909944 0.78 ADRA2A (0.49) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL8910486 0.77 ADRA2A (0.55) ADRA2AADRA2BADRA2CADRA1DADRA1A
Hydrochloric Acid SCHEMBL8909749 0.76 NPSR1 (0.50) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL8911033 0.76 ADRA2A (0.50) ADRA2AADRA2BADRA2CADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5639748-A HYPOTENSIVE AGENTS SMITHKLINE BEECHAM CORPORATION (US) 1997-06-17 US disclosed
EP-0630372-A1 HETEROALKOXY BENZAZEPINES SMITHKLINE BEECHAM CORPORATION (US) 1994-12-28 EP disclosed
EP-0630372-A4 HETEROALKOXY BENZAZEPINES. SMITHKLINE BEECHAM CORP (US) 1994-07-05 EP disclosed
WO-1993003015-A1 HETEROALKOXY BENZAZEPINES SMITHKLINE BEECHAM CORPORATION (US) 1993-02-18 WO disclosed