SCHEMBL8910294

SCHEMBL8910294

CCCC(CC)OP(=O)(O)Cc1nc(C2CCC2)cs1

nearest known ligand 0.32

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.31
HSD17B10 Q99714 2/20 0.30
ALOX15 P16050 1/20 0.30
CCR5 P51681 1/20 0.30
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
TP53 P04637 1/20 0.30
ADRB1 P08588 1/20 0.30
CYP3A4 P08684 1/20 0.30
ADORA3 P0DMS8 1/20 0.30
MAPT P10636 1/20 0.30
HPGD P15428 1/20 0.30
PTGS1 P23219 1/20 0.30
KMT2A Q03164 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8909270 0.85 RORC (0.32) RORC
SCHEMBL3818188 0.63 FDPS (0.44)
SCHEMBL22904608 0.62 MAPT (0.42) RORCHSD17B10ALOX15MEN1ALDH1A1
SCHEMBL11337222 0.61 FDPS (0.33) SMN1; SMN2
SCHEMBL3361922 0.60 RORC (0.41) RORCCCR5MAPTHPGDSMN1; SMN2
SCHEMBL75908 0.60 SMPD1 (0.48)
SCHEMBL11736280 0.60 PPARD (0.47)
SCHEMBL13043115 0.58 FDPS (0.43)
Hydrochloric Acid SCHEMBL11037597 0.58 SMPD1 (0.47)
SCHEMBL22204347 0.58 SMPD1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5637720-A Intermediate for (E)-4-[[3-[2-(4-cycloalkyl-2-thiazolyl)ethenyl]phenyl]amino-2,2-alkyldiyl-4-oxobutanoic acids HOFFMANN-LA ROCHE INC. (US) 1997-06-10 US disclosed
WO-1996008479-A1 A PROCESS OF MAKING (E)-4-[3-[2-(4-CYCLOALKYL-2-THIAZOLYL)ETHENYL]PHENYL]AMINO-2,2-ALKYLDIYL-4-OXOBUTANOIC ACID F. HOFFMANN-LA ROCHE AG (CH) 1996-03-21 WO disclosed