SCHEMBL8910495

SCHEMBL8910495

COc1ccccc1CNc1nc(Cl)nc2c1ncn2[C@@H]1O[C@H](CO)C(O)C1O

nearest known ligand 0.77

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NT5E P21589 2/20 0.65
ADORA3 P0DMS8 5/20 0.65
ADORA2A P29274 5/20 0.65
ADORA1 P30542 4/20 0.65
ADORA2B P29275 1/20 0.65
TSHR P16473 1/20 0.60
NFKB1 P19838 1/20 0.60
STAT6 P42226 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL743588 1.00 NT5E (0.65) NT5EADORA3ADORA2AADORA1ADORA2B
SCHEMBL743589 1.00 NT5E (0.65) NT5EADORA3ADORA2AADORA1ADORA2B
SCHEMBL774632 0.93 ADORA3 (0.64) NT5EADORA3ADORA2AADORA1ADORA2B
SCHEMBL742098 0.93 ADORA3 (0.64) NT5EADORA3ADORA2AADORA1ADORA2B
SCHEMBL740871 0.93 ADORA3 (0.64) NT5EADORA3ADORA2AADORA1ADORA2B
SCHEMBL742097 0.93 ADORA3 (0.64) NT5EADORA3ADORA2AADORA1ADORA2B
SCHEMBL638390 0.90 PGK1 (0.66) ADORA3ADORA2AADORA1ADORA2BTSHR
SCHEMBL638391 0.90 PGK1 (0.66) ADORA3ADORA2AADORA1ADORA2BTSHR
SCHEMBL743413 0.90 ADORA2A (0.61) ADORA3ADORA2AADORA1ADORA2BTSHR
SCHEMBL743414 0.90 ADORA2A (0.61) ADORA3ADORA2AADORA1ADORA2BTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0603348-A1 PURINE DERIVATIVES NOVO NORDISK A/S (DK) 1994-06-29 EP claimed
WO-1993023418-A1 PURINE DERIVATIVES NOVO NORDISK A/S (DK) 1993-11-25 WO claimed
US-5672588-A Purine derivatives NOVO NORDISK A/S (DK) 1997-09-30 US disclosed
EP-0603348-A1 PURINE DERIVATIVES NOVO NORDISK A/S (DK) 1994-06-29 EP disclosed
WO-1993023418-A1 PURINE DERIVATIVES NOVO NORDISK A/S (DK) 1993-11-25 WO disclosed