SCHEMBL8910904

SCHEMBL8910904

[CH2]C(c1ccc(N(C)C)cc1)c1ccc(N(C)C)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.58
TSHR P16473 6/20 0.58
HSD17B10 Q99714 3/20 0.58
ALOX15 P16050 2/20 0.58
SLC2A1 P11166 2/20 0.48
MAPK1 P28482 5/20 0.46
TDP1 Q9NUW8 4/20 0.46
CYP3A4 P08684 3/20 0.46
TP53 P04637 2/20 0.46
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.44
MAPT P10636 2/20 0.44
CYP1A2 P05177 1/20 0.44
PHLPP2 Q6ZVD8 1/20 0.44
RELA Q04206 1/20 0.43
GAA P10253 1/20 0.42
KDM4E B2RXH2 1/20 0.41
HPGD P15428 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9180847 0.93 ALDH1A1 (0.50) ALDH1A1TSHRHSD17B10ALOX15SLC2A1
SCHEMBL4074032 0.80 ALDH1A1 (0.52) ALDH1A1TSHRHSD17B10ALOX15SLC2A1
SCHEMBL61574 0.78 SLC2A1 (0.71) ALDH1A1TSHRHSD17B10ALOX15SLC2A1
SCHEMBL9626237 0.78 SLC2A1 (0.71) ALDH1A1TSHRHSD17B10ALOX15SLC2A1
SCHEMBL27270201 0.77 ALDH1A1 (0.48) ALDH1A1TSHRHSD17B10ALOX15SLC2A1
SCHEMBL65261 0.76 ALDH1A1 (1.00) ALDH1A1TSHRHSD17B10ALOX15SLC2A1
SCHEMBL346292 0.76 ALDH1A1 (0.61) ALDH1A1TSHRHSD17B10ALOX15SLC2A1
SCHEMBL10145543 0.76 ALDH1A1 (0.61) ALDH1A1TSHRHSD17B10ALOX15SLC2A1
SCHEMBL3893552 0.76 ALDH1A1 (0.61) ALDH1A1TSHRHSD17B10ALOX15SLC2A1
SCHEMBL61350 0.75 SLC2A1 (0.61) ALDH1A1TSHRHSD17B10ALOX15SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5622953-A DRUG RESISTANT TO ANTICANCER CHEMOTHERAPEUTIC DRUG BASF AKTIENGESELLSCHAFT (DE) 1997-04-22 US disclosed
EP-0691962-A1 1-AMINO-3-PHENOXY PROPANE DERIVATIVES AS MODULATORS OF MULTI-DRUG RESISTANCE BASF AKTIENGESELLSCHAFT (DE) 1996-01-17 EP disclosed
WO-1994022842-A1 1-AMINO-3-PHENOXY PROPANE DERIVATIVES AS MODULATORS OF MULTI-DRUG RESISTANCE BASF AKTIENGESELLSCHAFT (DE) 1994-10-13 WO disclosed