SCHEMBL8911265

SCHEMBL8911265

CCOC(=O)c1cccc2ncc(-c3ccccc3)cc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.53
MAPT P10636 6/20 0.53
SMN1; SMN2 Q16637 4/20 0.53
LMNA P02545 3/20 0.53
MAPK1 P28482 2/20 0.53
ATM Q13315 1/20 0.53
L3MBTL1 Q9Y468 3/20 0.53
KDM4E B2RXH2 2/20 0.53
TDP1 Q9NUW8 1/20 0.53
TP53 P04637 2/20 0.52
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
RXFP1 Q9HBX9 1/20 0.52
MEN1 O00255 1/20 0.51
PKM P14618 1/20 0.51
KMT2A Q03164 1/20 0.51
HPGD P15428 1/20 0.50
TSHR P16473 1/20 0.50
NMT1 P30419 2/20 0.49
NMT2 O60551 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8911758 0.85 AXL (0.62) ALDH1A1MAPTKDM4EMEN1KMT2A
SCHEMBL6421455 0.84 MAPT (0.55) ALDH1A1MAPTSMN1; SMN2MAPK1ATM
SCHEMBL10465583 0.83 ALDH1A1 (0.52) ALDH1A1MAPTSMN1; SMN2LMNAMAPK1
SCHEMBL28207288 0.81 MEN1 (0.58) ALDH1A1MAPTSMN1; SMN2LMNAMAPK1
SCHEMBL8912395 0.81 DHODH (0.49) ALDH1A1SMN1; SMN2LMNAKDM4ETP53
SCHEMBL8966261 0.80 PSMB5 (0.43) ALDH1A1MAPTSMN1; SMN2LMNAMAPK1
SCHEMBL2720141 0.79 ALDH1A1 (0.61) ALDH1A1MAPTSMN1; SMN2LMNAMAPK1
SCHEMBL9463382 0.79 NR3C2 (0.51) ALDH1A1MAPTSMN1; SMN2LMNAKDM4E
SCHEMBL31091353 0.79 ALDH1A1 (0.61) ALDH1A1MAPTSMN1; SMN2LMNAMAPK1
SCHEMBL9591718 0.79 ALDH1A1 (0.54) ALDH1A1MAPTSMN1; SMN2LMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5650514-A 3-substituted quinoline-5-carboxylic acid derivatives and processes for their preparation BAYER AKTIENGESELLSCHAFT (DE) 1997-07-22 US disclosed
US-5204472-A For preparing inotropic agents; substituted dihydropyridines BAYER AKTIENGESELLSCHAFT (DE) 1993-04-20 US disclosed
US-5100900-A Inotropic agents BAYER AKTIENGESELLSCHAFT (DE) 1992-03-31 US disclosed