SCHEMBL8911657

SCHEMBL8911657

CCCCCCC(C(=O)O)n1cnc2c(NC(=O)c3ccccc3-n3ncnn3)cccc21

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 1/20 0.42
AGTR2 P50052 1/20 0.42
ADA P00813 1/20 0.37
TDP1 Q9NUW8 3/20 0.36
PTPN1 P18031 3/20 0.35
HCRTR1 O43613 4/20 0.35
HCRTR2 O43614 4/20 0.35
CNR2 P34972 4/20 0.34
CNR1 P21554 2/20 0.34
PLK1 P53350 3/20 0.34
CASP1 P29466 1/20 0.33
PLK3 Q9H4B4 2/20 0.33
PTPN2 P17706 1/20 0.33
PTPN6 P29350 1/20 0.33
CDC25B P30305 1/20 0.33
PTPN11 Q06124 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7015254 0.78
SCHEMBL668253 0.69 ASAH1 (0.51) AGTR1AGTR2ADA
SCHEMBL9091629 0.64 AGTR1 (0.77) AGTR1AGTR2PTPN1PLK1PLK3
SCHEMBL9092112 0.62 AGTR1 (0.46) AGTR1AGTR2
SCHEMBL7020223 0.62 PTPN11 (0.43) AGTR1AGTR2PTPN11
SCHEMBL24476294 0.62 P2RX7 (0.41) ADA
SCHEMBL24476401 0.62 P2RX7 (0.41) ADA
SCHEMBL7016171 0.62
SCHEMBL9091837 0.62 AGTR1 (0.82) AGTR1AGTR2PLK1
Hydrochloric Acid SCHEMBL9087410 0.61 AGTR1 (0.58) AGTR1AGTR2PTPN1PLK1PLK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5612360-A AROMATIC N-HETEROCYCLIC COMPOUNDS AS HYPOTENSIVE AGENTS WITH ACID GROUPS, SULFONYLCARBOXAMIDES OR TETRAZOLE GROUPS ELI LILLY AND COMPANY (US) 1997-03-18 US disclosed