SCHEMBL8911804

SCHEMBL8911804

Fc1ccc(C2CCC3(CCC(c4cccc(C(F)(F)F)c4)CO3)OC2)cc1

nearest known ligand 0.64

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 6/20 0.64
HTR2C P28335 3/20 0.47
DRD2 P14416 1/20 0.41
HTR2A P28223 1/20 0.39
HTR2B P41595 1/20 0.39
HTR1A P08908 1/20 0.37
KDM1A O60341 1/20 0.36
RCOR1 Q9UKL0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8503079 0.87 TACR1 (0.61) TACR1HTR2CDRD2HTR2AHTR2B
SCHEMBL8502905 0.87 TACR1 (0.61) TACR1HTR2CDRD2HTR2AHTR2B
SCHEMBL22816111 0.81 HTR2C (0.57) TACR1HTR2CDRD2HTR2AHTR2B
SCHEMBL8504929 0.80 TACR1 (0.49) TACR1HTR2CDRD2
SCHEMBL8907338 0.80 HTR2C (0.52) TACR1HTR2CDRD2HTR2AHTR2B
SCHEMBL8907343 0.77 TACR1 (0.49) TACR1HTR2CDRD2HTR2AHTR2B
SCHEMBL1065758 0.71 HTR2C (0.77) HTR2CDRD2HTR2AHTR2BHTR1A
SCHEMBL744072 0.70 RAB9A (0.37) TACR1DRD2HTR2AHTR1AKDM1A
SCHEMBL22816650 0.69 HTR2C (0.53) TACR1HTR2CKDM1ARCOR1
SCHEMBL2427723 0.68 HTR2C (0.58) TACR1HTR2CDRD2HTR2AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799231-A1 SPIROKETAL DERIVATIVES, COMPOSITIONS CONTAINING THEM AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LTD. (GB) 1997-10-08 EP claimed