SCHEMBL8912015

SCHEMBL8912015

Cc1ccc([C@H](NC(=O)OC(C)(C)C)[C@@H](O)C(=O)O)cc1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 6/20 0.46
PPARG P37231 5/20 0.46
KEAP1 Q14145 5/20 0.43
NFE2L2 Q16236 5/20 0.43
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
ALDH1A1 P00352 2/20 0.40
TSHR P16473 1/20 0.40
LMNA P02545 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ATM Q13315 1/20 0.38
ACE P12821 1/20 0.38
HPGD P15428 1/20 0.37
PPARD Q03181 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6443317 0.89 PPARA (0.48) PPARAPPARGCTSSCTSKALDH1A1
SCHEMBL12070284 0.88 CTSK (0.51) PPARAPPARGCTSSCTSKATM
SCHEMBL7087412 0.88 CTSK (0.51) PPARAPPARGCTSSCTSKATM
SCHEMBL144832 0.88 CTSK (0.51) PPARAPPARGCTSSCTSKATM
SCHEMBL13363641 0.88 CTSK (0.51) PPARAPPARGCTSSCTSKATM
SCHEMBL335777 0.88 CTSK (0.51) PPARAPPARGCTSSCTSKATM
SCHEMBL767076 0.88 CTSK (0.51) PPARAPPARGCTSSCTSKATM
SCHEMBL6166 0.88 CTSK (0.51) PPARAPPARGCTSSCTSKATM
SCHEMBL8886861 0.88 CTSK (0.51) PPARAPPARGCTSSCTSKATM
SCHEMBL7625656 0.87 MAPT (0.46) PPARAPPARGCTSSCTSKATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008024299-A2 COMBINATION WITH BIS(THIOHYDRAZIDE AMIDES) FOR TREATING CANCER SYNTA PHARMACEUTICALS CORP. (US) 2008-02-28 WO disclosed
WO-2008024305-A2 BIS (THIOHYDRAZIDE AMIDES) FOR TREATING MELANOMA SYNTA PHARMACEUTICALS CORP. (US) 2008-02-28 WO disclosed
US-5606068-A Acid anhydrides, their preparation and their use RHONE-POULENC RORER S.A. (FR) 1997-02-25 US disclosed
US-5476954-A Condensing hydroxyl protected taxane derivative with oxazolidine derivative, decyclizing in acid medium, reacting butoxycarbonyl or benzoyl radical with amine, deprotecting, isolating, purifying product RHONE-POULENC RORER S.A. (FR) 1995-12-19 US disclosed