Oxalic Acid

Oxalic Acid

SCHEMBL8913669

CS(=O)(=O)Nc1ccc2c(c1)CC1(CCCN(CCc3ccc([N+](=O)[O-])cc3)C1)O2.O=C(O)C(=O)O

nearest known ligand 0.61

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

OPRM1SLC6A4

The experimentally established mechanism targets of Oxalic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.42
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
KCNJ1 P48048 1/20 0.41
HRH3 Q9Y5N1 1/20 0.40
ABCB1 P08183 2/20 0.39
ABCG2 Q9UNQ0 2/20 0.39
ADRA1D P25100 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8912442 0.96 KCNH2 (0.45) KCNH2HDAC3HDAC4HDAC1HDAC7
Oxalic Acid SCHEMBL8914314 0.92 KCNH2 (0.46) KCNH2HDAC3HDAC4HDAC1HDAC7
Oxalic Acid SCHEMBL8914466 0.89 KDM4E (0.49) HRH3
Oxalic Acid SCHEMBL8566135 0.77 HDAC3 (0.55) KCNH2HDAC3HDAC4HDAC1HDAC7
SCHEMBL8571720 0.76 KCNH2 (0.70) KCNH2ADRA1D
Hydrochloric Acid SCHEMBL8913401 0.75 ADRA1D (0.64) KCNH2ADRA1D
Hydrochloric Acid SCHEMBL8922961 0.75 KCNH2 (0.43) KCNH2ADRA1D
SCHEMBL8912969 0.73 HDAC3 (0.48) KCNH2HDAC3HDAC4HDAC1HDAC7
SCHEMBL8921191 0.68 DRD2 (0.56) KCNH2ADRA1D
SCHEMBL8914120 0.68 HDAC3 (0.47) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed
EP-0431943-A2 Nitrogen-containing spirocycles MERCK & CO. INC. (US) 1991-06-12 EP disclosed